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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T36949 Niaprazine 27367-90-4 98%
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for s...
T12444 Phentolamine Analogue 1 47142-51-8 98%
Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.
T2547 Droxidopa 23651-95-8 98%
Droxidopa (L-DOPS) is an orally available prodrug of norepinephrine that is used in the treatment of symptomatic orthostatic hypotension due to neurogenic causes...
T22904 L-745870 trihydrochloride 866021-03-6 98%
L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.
T8663 Nifenalol.HCl 5704-60-9 98%
Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.
T0948 Adrenalone hydrochloride 62-13-5 98%
Adrenalone hydrochloride (Adrenalone HCl) is a dopamine β-oxidase inhibitor with a similar structure to the norepinephrine transporter (NET) ligand, with an IC50...
T1066L Ketanserin tartrate 83846-83-7 98%
Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist with antihypertensive activity, inhibits serotonin-induced vaso...
T83965 Tamsolusin Hydrochloride 80223-99-0 98%
Tamsolusin Hydrochloride (YM 12617) is a highly selective alpha-1A adrenergic receptor antagonist used in the treatment of benign prostatic hypertrophy.
T11607 ICI 118,551 hydrochloride 72795-01-8 98%
ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3 recep...
T5954 Methyldopa hydrate 41372-08-1
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sym...
T7164 Levalbuterol tartrate 661464-94-4
Levalbuterol tartrate (Levosalbutamol tartrate) is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
T0248 Clorprenaline hydrochloride 6933-90-0
Clorprenaline hydrochloride (Clorprenaline HCl) is a beta-2 adrenergic agonist with bronchodilator activity.
T6662 Scopine 498-45-3
Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
T0317 Buflomedil hydrochloride 35543-24-9
Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.
T0348 Labetalol hydrochloride 32780-64-6
Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
T0165 Urapidil 34661-75-1
Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
T1064 Norepinephrine bitartrate monohydrate 108341-18-0
Norepinephrine bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator.
T0394 Moxisylyte hydrochloride 964-52-3
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
T6765 Atipamezole hydrochloride 104075-48-1
Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochlor...
T5028 Landiolol hydrochloride 144481-98-1
Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.
Niaprazine
T36949
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for s...
Phentolamine Analogue 1
T12444
Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.
Droxidopa
T2547
Droxidopa (L-DOPS) is an orally available prodrug of norepinephrine that is used in the treatment of symptomatic orthostatic hypotension due to neurogenic causes...
L-745870 trihydrochloride
T22904
L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.
nifenalol.HCl
T8663
Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.
Adrenalone hydrochloride
T0948
Adrenalone hydrochloride (Adrenalone HCl) is a dopamine β-oxidase inhibitor with a similar structure to the norepinephrine transporter (NET) ligand, with an IC50...
Ketanserin tartrate
T1066L
Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist with antihypertensive activity, inhibits serotonin-induced vaso...
Tamsolusin Hydrochloride
T83965
Tamsolusin Hydrochloride (YM 12617) is a highly selective alpha-1A adrenergic receptor antagonist used in the treatment of benign prostatic hypertrophy.
ICI 118,551 hydrochloride
T11607
ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3 recep...
Methyldopa hydrate
T5954
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sym...
Levalbuterol tartrate
T7164
Levalbuterol tartrate (Levosalbutamol tartrate) is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
Clorprenaline hydrochloride
T0248
Clorprenaline hydrochloride (Clorprenaline HCl) is a beta-2 adrenergic agonist with bronchodilator activity.
Scopine
T6662
Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
Buflomedil hydrochloride
T0317
Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.
Labetalol hydrochloride
T0348
Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
Urapidil
T0165
Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
Norepinephrine bitartrate monohydrate
T1064
Norepinephrine bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator.
Moxisylyte hydrochloride
T0394
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
Atipamezole hydrochloride
T6765
Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochlor...
Landiolol hydrochloride
T5028
Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.
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