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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T6600 Naftopidil dihydrochloride 57149-08-3 98%
Naftopidil DiHCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
T6653 Salmeterol Xinafoate 94749-08-3 98%
Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstruc...
T21445 Naphazoline 835-31-4 98%
Naphazoline is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in reducing swe...
T16759 Ritanserin 87051-43-2 98%
Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adren...
T22406 Prazosin 19216-56-9 98%
Prazosin, an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
T3232 Higenamine hydrochloride 11041-94-4 98%
Higenamine(Hydrochloride) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein–coupl...
T0154 Nebivolol hydrochloride 152520-56-4 98%
Nebivolol hydrochloride is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR through the endothelial L-argin...
T36949 Niaprazine 27367-90-4 98%
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for s...
T3158 Harmane 486-84-0 98%
Harmane is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
T5954 Methyldopa hydrate 41372-08-1 98%
Alpha-Methyldopa Sesquihydrate is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sympathe...
T6522 Guanabenz Acetate 23256-50-0 98%
Guanabenz Acetate is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor is 8.2...
T6641 Rilmenidine Phosphate 85409-38-7 98%
Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.
T22245 Arformoterol Tartrate 200815-49-2 98%
Arformoterol Tartrate is the tartrate salt of arformoterol. Arformoterol is a long-acting beta-2 adrenergic agonist with bronchodilator activity[2].
T19680 Zotepine 26615-21-4 98%
Zotepine is a second-generation antipsychotic with a primary use as a treatment for schizophrenia, although clinical trials have been conducted into its efficacy...
T1275 Phentolamine mesylate 65-28-1 98%
Phentolamine mesylate is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma, ...
T7164 Levalbuterol tartrate 661464-94-4 98%
Levosalbutamol tartrate is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
T0696 Naftopidil 57149-07-2 98%
Naftopidil (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
T0226 Betaxolol hydrochloride 63659-19-8 98%
Betaxolol is a cardioselective beta-blocker used in the treatment of hypertension. Betaxolol has not been linked to instances of clinically apparent drug induced...
T12444 Phentolamine Analogue 1 47142-51-8 98%
Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.
T0324 Isoxsuprine hydrochloride 579-56-6 98%
Isoxsuprine hydrochloride is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
Naftopidil dihydrochloride
T6600
Naftopidil DiHCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
Salmeterol Xinafoate
T6653
Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstruc...
Naphazoline
T21445
Naphazoline is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in reducing swe...
Ritanserin
T16759
Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adren...
Prazosin
T22406
Prazosin, an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
Higenamine hydrochloride
T3232
Higenamine(Hydrochloride) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein–coupl...
Nebivolol hydrochloride
T0154
Nebivolol hydrochloride is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR through the endothelial L-argin...
Niaprazine
T36949
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for s...
Harmane
T3158
Harmane is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
Methyldopa hydrate
T5954
Alpha-Methyldopa Sesquihydrate is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sympathe...
Guanabenz Acetate
T6522
Guanabenz Acetate is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor is 8.2...
Rilmenidine Phosphate
T6641
Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.
Arformoterol Tartrate
T22245
Arformoterol Tartrate is the tartrate salt of arformoterol. Arformoterol is a long-acting beta-2 adrenergic agonist with bronchodilator activity[2].
Zotepine
T19680
Zotepine is a second-generation antipsychotic with a primary use as a treatment for schizophrenia, although clinical trials have been conducted into its efficacy...
Phentolamine mesylate
T1275
Phentolamine mesylate is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma, ...
Levalbuterol tartrate
T7164
Levosalbutamol tartrate is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
Naftopidil
T0696
Naftopidil (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
Betaxolol hydrochloride
T0226
Betaxolol is a cardioselective beta-blocker used in the treatment of hypertension. Betaxolol has not been linked to instances of clinically apparent drug induced...
Phentolamine Analogue 1
T12444
Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.
Isoxsuprine hydrochloride
T0324
Isoxsuprine hydrochloride is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
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