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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T24257 | KCA-1490 | KCA 1490,KCA1490 | |
KCA-1490 is an inhibitor of dual PDE3/4. | |||
T15647 | Tipelukast | MN 001,KCA 757 | Leukotriene Receptor |
Tipelukast (KCA 757) is a novel orally available leukotriene receptor antagonist with anti-inflammatory activity that reduces fibrosis and down-regulates TIMP-1, type 1 collagen.Tipelukast is used in the study of asthma. | |||
T1449 | Hydrochlorothiazide | HCTZ | Potassium Channel , Carbonic Anhydrase , TGF-beta/Smad |
Hydrochlorothiazide (HCTZ) is a Thiazide Diuretic. The physiologic effect of hydrochlorothiazide is by means of Increased Diuresis. | |||
T60985 | KCa2 channel modulator 1 | ||
KCa2 channel modulator 1 (compound 2o) is an effective subtype-selective K/Ca2 channel positive modulator that potentiates rat K Ca 2.2 channel subtype with an EC 50 value of 0.99 μM and human K Ca 2.3 channels subtype w... | |||
T60986 | KCa2 channel modulator 2 | ||
KCa2 channel modulator 2 (compound 2q) is an effective subtype-selective K/Ca 2 channel positive modulator which shows similar potency on the human K Ca 2.3 channel and rat K Ca 2.2a subtypes, with EC50 values of 0.60 μM... | |||
T72195 | KCa1.1 channel activator-2 | ||
KCa1.1 channel activator-2, a hybrid derivative of Quercetin, selectively stimulates the vascular KCa1.1 channels. This compound demonstrates significant myorelaxant activity. | |||
T72194 | KCa1.1 channel activator-1 | ||
KCa1.1 Channel Activator-1, a hybrid derivative of Quercetin, selectively stimulates the vascular KCa1.1 channels while also blocking CaV1.2 channels. Additionally, it demonstrates weak myorelaxant activity. | |||
T76184 | Scyllatoxin | ||
Scyllatoxin (Leiurotoxin I), a peptide toxin derived from the venom of the scorpion (Leiurus quinquestriatus hebraeus), acts as a blocker of small-conductance K Ca (SK) channels. It notably enhances the release of norepi... |