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Search Results for " LDK378 "

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カタログ番号 製品名 別名 ターゲット
T1791 Ceritinib LDK378 Serine Protease , IGF-1R , ALK
Ceritinib (LDK378) is a specific ALK inhibitor (IC50: 0.2 nM).
T1791L Ceritinib dihydrochloride LDK378 dihydrochloride IGF-1R , ALK
Ceritinib dihydrochloride (LDK378 dihydrochloride) is a selective, orally bioavailable and ATP-competitive inhibitor of ALK tyrosine kinase(IC50 of 200 pM), and also inhibits IGF-1R, InsR, and STK22D (IC50 values of 8, 7...
T10766 Ceritinib D7 LDK378 D7 Others
Ceritinib D7 (LDK378 D7) is a deuterium-labeled Ceritinib. Ceritinib is an ATP-competitive inhibitor of ALK tyrosine kinase.