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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T21337 | Lurasidone | SM-13496 | Dopamine Receptor , 5-HT Receptor |
Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6.75 nM). | |||
T1735 | Lurasidone hydrochloride | Lurasidone HCl,SM-13496 (Hydrochloride),SM-13496 | Dopamine Receptor , 5-HT Receptor , Norepinephrine |
Lurasidone hydrochloride (Lurasidone HCl) is a thiazole derivative and atypical antipsychotic agent that functions as a dopamine D2 receptor antagonist; serotonin 5-HT2 receptor antagonist, serotonin 5-HT7 receptor antag... | |||
T11893L | Lurasidone metabolite 14326 hydrochloride | Lurasidone metabolite 14326 hydrochloride (186204-33-1 free base) | Others |
Lurasidone metabolite 14326 hydrochloride, an active metabolite of the atypical antipsychotic Lurasidone, maintains its significant function in pharmacological efficacy. | |||
TMIH-0315 | Lurasidone Inactive Metabolite 14283-d8 | 5α/6α-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers) | |
Lurasidone Inactive Metabolite 14283-d8 is a deuterated compound of Lurasidone Inactive Metabolite 14283.Lurasidone Inactive Metabolite 14283 has a CAS number of 186204-31-9. | |||
TMIH-0316 | Lurasidone Inactive Metabolite 14326-d8 | 5β/6β-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers) | |
Lurasidone Inactive Metabolite 14326-d8 is a deuterated compound of Lurasidone Inactive Metabolite 14326.Lurasidone Inactive Metabolite 14326 has a CAS number of 186204-33-1. | |||
T11893 | Lurasidone metabolite 14326 | Others | |
Lurasidone metabolite 14326, an active metabolite of the atypical antipsychotic Lurasidone, functions effectively in the body. | |||
T13760 | Lurasidone Metabolite 14283 hydrochloride | Others | |
Lurasidone Metabolite 14283 hydrochloride is a major active metabolite of Lurasidone. | |||
T19407 | Lurasidone Metabolite 14326 D8 | Others | |
Lurasidone Metabolite 14326 D8 is the deuterium labeled Lurasidone Metabolite 14326. | |||
T11892 | Lurasidone D8 Hydrochloride | SM-13496 D8 | Others |
Lurasidone D8 Hydrochloride is an inhibitor of Dopamine D2, 5-HT2A, 5-HT7, 5-HT1A and noradrenaline α2C, and is the deuterium labeled Lurasidone. | |||
T19406 | Lurasidone Metabolite 14283 D8 | Others | |
Lurasidone Metabolite 14283 D8 is the deuterium labeled Lurasidone Metabolite 14283. | |||
TMIH-0313 | lurasidone-d8 | ||
lurasidone-d8 is a deuterated compound of lurasidone. | |||
TMIH-0314 | Lurasidone-d8 HCl | ||
Lurasidone-d8 HCl is a deuterated compound of Lurasidone HCl. Lurasidone HCl has a CAS number of 367514-88-3. Lurasidone hydrochloride is a thiazole derivative and atypical antipsychotic agent that functions as a dopamin... |