8
2
1
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T60002 | DC-S239 | Histone Methyltransferase | |
DC-S239 (DC-S239) is a selective inhibitor of histone methyltransferase SETD7 (IC50 = 4.59 μM) with anticancer activity. | |||
T10682L | CARM1-IN-1 | CARM1-IN-7G | Histone Methyltransferase |
CARM1-IN-1 (CARM1-IN-7G) is a selective inhibitor of CARM1 with IC50 of 8.6 μM. CARM1-IN-1 shows weak activity against PRMT1 and SET7 with IC50 > 600 μM. | |||
T16886 | Sinefungin | Adenosyl-Ornithine,A-9145,Antibiotic 32232RP | Others , Histone Methyltransferase , Antibiotic , Antifungal |
Sinefungin (Adenosyl-Ornithine) is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viral multiplication. Sinefungin is a SET7/9 inhibitor and ameliorates r... | |||
T68613 | DC-S238 | ||
DC-S238 is a potent and selective histone methyltransferase SET7 inhibitor. | |||
T71918 | DC-S100 | ||
DC-S100 is a selective histone methyltransferase SET7 inhibitor. | |||
T72013 | Epigenetic Multiple Ligand | ||
Epigenetic Multiple Ligand is a cell-permeable inhibitor of substrate processing by several chromatin-associated enzymes, including SIRT1/2, H3/SET7, H3/p300/CBP, H4/RmtA, PABP1/CARM1, and H4/PRMT1. It acts by inducing e... | |||
T26188 | Setin-1 | ||
Setin-1 is the most potent Set7 inhibitor that acts by inhibiting the KMTase G9a. | |||
T64186 | CARM1-IN-1 hydrochloride | ||
CARM1-IN-1 hydrochloride is a potent and selective inhibitor of CARM1 (IC50: 8.6 μM) with low inhibition of PRMT1 and SET7. |
カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPY-01584 | PR-Set7 Protein, Human, Recombinant | Human | E. coli |
KMT5A (known as PR-Set7/9, SETD8 and SET8), a member of the SET domain containing methyltransferase family specifically targeting H4K20 for methylation, has been implicated in multiple biological processes. Inhibition of... | |||
TMPY-01229 | SETD7 Protein, Human, Recombinant (His) | Human | E. coli |
Histone-lysine N-methyltransferase SETD7, also known as SET domain containing (lysine methyltransferase) 7, SET7/9, Histone H3-K4 methyltransferase SETD7, H3-K4-HMTase SETD7, and SETD7, is a member of the histone-lysine ... |
カタログ番号 | 製品名 | ||
---|---|---|---|
L2191 | Anti-Breast Cancer Compound Library | 1939 compounds | |
A unique collection of 1939 compounds with anti-breast cancer therapeutic activity or targeting breast cancer’s major signaling pathways, can be used for anti-breast cancer drug discovery and mechanism study; |