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TP2207 |
Pasireotide Acetate
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Somatostatin
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Pasireotide Acetate is a stable cyclohexapeptide somatostatin mimic |
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TP1570L |
Cortistatin-14 acetate
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Cortistatin-14 acetate(186901-48-4 Free base) |
Somatostatin
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Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5). Cortistatin-14 acetate shows anticonvulsive, neuroprotective... |
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TP1346 |
CYN 154806 TFA
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CYN 154806 TFA |
Somatostatin
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CYN 154806 TFA is a cyclic octapeptide and an effective selective somatostatin sst2 receptor antagonist. For the recombinant sst2, sst1, sst3, sst4 and sst5 receptors, the pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48... |
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T23479 |
TT 232
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Others
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sst1/sst4 somatostatin receptors agonist |
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TP2045 |
CH 275
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Potent somatostatin receptor 1 (sst1) agonist; displays selectivity for sst1 (IC50 values are 30.9 nM, 345 nM, > 1 μM, > 10 μM and > 10μM for human sst1, sst3, sst4, sst2 and sst5 respectively). Attenuates somatostatin r... |
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T12368 |
Pasireotide L-aspartate salt
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SOM230 L-aspartate |
Others
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Pasireotide L-aspartate salt is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9 respectively). |
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T76034 |
Cortistatin-14 TFA
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Cortistatin-14 (TFA), a neuropeptide resembling somatostatin-14 in structure, operates through interaction with somatostatin receptors (sst1-sst5). This compound exhibits anticonvulsive and neuroprotective effects alongs... |
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T32511L |
L-796,778 acetate
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L-796,778 acetate(217480-25-6 Free base) |
Somatostatin
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L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM. |
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TP1877 |
CYN 154806
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CYN 154806 is a potent and selective somatostatin sst2 receptor antagonist, The pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively. |
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T12370 |
Pasireotide
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SOM 230,SOM 320 |
Others
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Pasireotide(SOM 230) is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9 respectively). |
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TP2122 |
Seglitide
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Peptide agonist for sst2 and sst5 somatostatin receptors. IC50/Kd values (nM) at cloned human somatostatin receptors are: > 1000 (sst1), 0.2 - 1.5 (sst2), 27 - 36 (sst3), > 127 (sst4), and 0.06 - 23 (sst5). |
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T75248 |
Pasireotide (diaspartate)
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Pasireotide diaspartate (SOM230), a long-acting cyclohexapeptide and somatostatin analog, enhances agonist activity across somatostatin receptor subtypes (sst1/2/3/4/5, with pK i values of 8.2, 9.0, 9.1, <7.0, and 9.9, r... |
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T28851 |
SRA880 free base
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SRA 880,NVPSRA880,NVP SRA880,NVP-SRA880,SRA-880,SRA880 |
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SRA880 is a non-peptide antagonist of somatostatin sst1-receptor. SRA880 displayed significantly lower affinity for the other human recombinant somatostatin receptors ( pK(d) < or = 6.0). SRA880 shows a certain binding a... |
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T35663 |
Cortistatin-29 (rat) (trifluoroacetate salt)
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Cortistatin-29 is a neuropeptide that is structurally similar to somatostatin-28. It is produced by cleavage of preprocortistatin to procortistatin, which is cleaved at dibasic amino acids to form cortistatin-29 and cort... |
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T76596 |
PRL 3195
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PRL 3195 is a somatostatin receptor antagonist, exhibiting K i values of 6, 17, 66, 1000, and 1000 nM for human somatostatin receptors sst 5 , sst 2 , sst 3 , sst 1 , and sst 4, respectively [1]. |
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T11800 |
L-803087
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Somatostatin
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T12369 |
Pasireotide pamoate
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SOM230 pamoate |
Others
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Pasireotide pamoate is a stable cyclohexapeptide somatostatin mimic. Pasireotide pamoate exhibits antisecretory, antiproliferative, and proapoptotic activity. |
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T13811 |
Pasireotide ditrifluoroacetate
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SOM230 ditrifluoroacetate,Pasireotide ditrifluoroacetate (396091-73-9 free base),Pasireotide TFA salt |
Others
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Pasireotide is a stable cyclohexapeptide somatostatin mimic. |
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T39207 |
L-803087 TFA
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L-803087 TFA is a highly potent and selective agonist of the somatostatin sst4 receptor, exhibiting a Ki value of 0.7 nM. It displays a remarkable selectivity, being over 280-fold more preferential for the sst4 receptor ... |
