Glucagon Receptor

The glucagon receptor is a 62 kDa protein that is activated by glucagon and is a member of the class B G-protein coupled family of receptors, coupled to G alpha i, Gs and to a lesser extent G alpha q. Stimulation of the receptor results in activation of adenylate cyclase and increased levels of intracellular cAMP. In humans, the glucagon receptor is encoded by the GCGR gene.

Cat. No.	製品名	CAS No.	Purity
T9579L	GLP-1 receptor agonist 9 citrate	T9579L	98%
T9579L	GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
T19117	3-Deoxyglucosone	4084-27-9	98%
T19117	3-Deoxyglucosone(3-Deoxy-D-glucosone) is synthesized by the intermediate pathway of the melad and polyol reactions.3-Deoxyglucosone reacts rapidly with protein a...
T9579	GLP-1 receptor agonist 9	2401892-71-3	98%
T9579	1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
T15387	GLP-1R Antagonist 1	488097-06-9	98%
T15387	GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).
T35337L	Teduglutide acetate		98%
T35337L	Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy. Teduglutide acetate partially restores small intestinal epithelial functio...
TP1976L	Oxyntomodulin acetate		98%
TP1976L	Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
TP2252	GLP-1 (9-36) amide	161748-29-4	98%
TP2252	antagonist at the human GLP-1 receptor
TP1039	Secretin (33-59), rat	121028-49-7	98%
TP1039	Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.
TP1863L	Glucagon (19-29), human acetate	TP1863L	98%
TP1863L	Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.
T37890L	GLP-1(28-36)amide acetate	T37890L	98%
T37890L	GLP-1(28-36)amide acetate inhibits mitochondrial permeability transition with antioxidant, anti-diabetic and cardioprotection activities.
TP2100L	Avexitide acetate	2051593-46-3	98%
TP2100L	Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.
TP2100	Avexitide	133514-43-9
TP2100	Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.
TP1419L	HAEGTFT acetate(926018-95-3 free base)	TP1419L	100%
TP1419L	HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
TP1796	Albiglutide TFA (782500-75-8 free base)	TP1796	100%
TP1796	Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
T60047L	V-0219 hydrochloride	T60047L	100%
T60047L	V-0219 hydrochloride, an orally-active positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R), is utilized in obesity-associated di...
T22893	L-168049	191034-25-0	100%
T22893	L-168049 is a selective and non-competitive antagonist of human glucagon receptor with IC50s of 3.7 nM, 63 nM, and 60 nM for human, murine, and canine, respectiv...
T63909	GLP-1R agonist 3	2428640-18-8	97.19%
T63909	GLP-1R agonist 3 is a thickened imidazole derivative compound that is a potent agonist of GLP-1R. GLP-1R agonist 3 has shown research potential in diabetes.
TP1111L	Tirzepatide Acetate(2023788-19-2 free base)	TP1111L	97.3%
TP1111L	Tirzepatide acetate is a dual GIP / GLP-1 receptor agonist.
T3422	GRA Ex-25	307983-31-9	97.39%
T3422	GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.
TP1382L	HAEGTFTSDVS acetate	TP1382L	97.47%
TP1382L	HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.