ペプチド
抗体
色素試薬
PROTAC
バーチャルスクリーニング
TargetMolキット
Cell Counting Kit-8 (CCK-8)
Inhibitor Cocktails
天然化合物
フェノール類
アルカロイド類
フラボノイド類
阻害剤
血管新生
アポトーシス
オートファジー
細胞周期・チェックポイント
クロマチン・エピジェネティック
細胞骨格シグナル
DNA損傷・DNA修復
内分泌・ホルモン
GPCR/Gタンパク質
免疫・炎症
JAK・STATシグナル
| Cat. No. | 製品名 | CAS No. | Purity | Chemical Structure |
|---|---|---|---|---|
| T9256 | N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine | 1071135-06-2 | 98% |
|
| N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine is a novel 2,6-naphthyridine identified by high throughput screen (HTS) as a dual protein... | ||||
| T1808 | Kb-NB77-78 | 1350622-33-1 | 98% |
|
| kb-NB77-78 is an analog of CID797718, which is a by-product of the synthesis of the parental compound, CID755673(PKD1 inhibitor). | ||||
| T1858 | CID-797718 | 370586-05-3 | 98% |
|
| CID797718 is a protein kinase D1 (PKD1) inhibitor. | ||||
| T15781 | LP-935509 | 1454555-29-3 | 98% |
|
| LP-935509 is highly brain-penetrant and reverses fully established pain behavior following the SNL procedure. LP-935509 is also an effective inhibitor of BIKE (I... | ||||
| T77501 | TAO Kinase inhibitor 2 | 850467-77-5 | 98% |
|
| TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM. | ||||
| T1863 | CID 2011756 | 638156-11-3 | 98% |
|
| CID-2011756 is an ATP-competitive and specific PKD1 inhibitor. | ||||
| T4058 | R-IMPP | 2133832-83-2 | 98% |
|
| R-IMPP is an inhibitor of PCSK9 translation. R-IMPP stimulates uptake of LDL-C in hepatoma cells by increasing LDL-R levels, without altering levels of secreted ... | ||||
| T8676 | FOY 251 | 71079-09-9 | 98% |
|
| FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate. | ||||
| T1954 | SRPIN340 | 218156-96-8 | 98% |
|
| SRPIN340, a serine/arginine-rich protein kinase (SRPK)-specific inhibitor, is potent for SRPK1 (IC50 = 0.89 uM). | ||||
| T3060 | Fasudil hydrochloride | 105628-07-7 | 98% |
|
| Fasudil Hydrochloride is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki of 0.33 μM, 1.0 μM, 9.3 μM and 55 μM, respectively. | ||||
| T1606 | Fasudil | 103745-39-7 | 98% |
|
| Fasudil is a potent inhibitor of ROCK1, PKA, PKC, and MLCK. | ||||
| T8957L | CRT0066101 dihydrochloride(956121-30-5 free base) | 2308510-39-4 | 98% |
|
| CRT0066101 dihydrochloride is an inhibitor of PKD. | ||||
| T2062 | Kb NB 142-70 | 1233533-04-4 | 98% |
|
| kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively). | ||||
| T5456 | WNK-IN-11 | 2123489-30-3 | 98% |
|
| WNK-IN-11 is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM) | ||||
| T7017 | WNK463 | 2012607-27-9 | 98% |
|
| WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4). | ||||
| T11666 | IPR-803 | 892243-35-5 | 98% |
|
| IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity. IPR-803 binds directly to uPAR with a Ki of 0.2 μM.... | ||||
| T2626 | SBC-115076 | 489415-96-5 | 98% |
|
| SBC-115076 is a potent extracellular proprotein convertase subtilisin kexin type 9 (PCSK9) antagonist. | ||||
| T2392 | Nafamostat mesylate | 82956-11-4 | 98% |
|
| Nafamostat mesylate, a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitis and atopic de... | ||||
| T10547 | BioE-1115 | 1268863-35-9 | 98% |
|
| BioE-1115 is a selective and potent inhibitor of serine-threonine protein kinase (PASK, IC50 = 4 nM). BioE-1115 is a potent inhibitor of CK2α (IC50 = 10 μM). | ||||
| T19763 | Cetraxate hydrochloride | 27724-96-5 | 98% |
|
| Cetraxate HCl is an oral gastrointestinal medication. It has a cytoprotective effect. | ||||
