Powder: -20°C for 3 years | In solvent: -80°C for 1 year
AZ10606120 dihydrochloride is a selectable, potent, high-affinity receptor antagonist with K D values of 1.4 and 19 nM at human and rat P2X 7 receptors, respectively. AZ10606120 dihydrochloride inhibits tumor growth and has anti-angiogenic activity. AZ 10606120 acts as a negative allosteric modulator when bound to a site coupled to the ATP binding site.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 14,000 |
5 mg | 在庫あり | ¥ 34,000 |
10 mg | 在庫あり | ¥ 55,000 |
25 mg | 在庫あり | ¥ 110,000 |
50 mg | 約6-8 週間 | ¥ 158,000 |
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 37,500 |
説明 | AZ10606120 dihydrochloride is a selectable, potent, high-affinity receptor antagonist with K D values of 1.4 and 19 nM at human and rat P2X 7 receptors, respectively. AZ10606120 dihydrochloride inhibits tumor growth and has anti-angiogenic activity. AZ 10606120 acts as a negative allosteric modulator when bound to a site coupled to the ATP binding site. |
ターゲット&IC50 | P2X7:10 nM |
分子量 | 495.48 |
分子式 | C25H36Cl2N4O2 |
CAS No. | 607378-18-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 8 mg/mL (16.15 mM), Sonication is recommended.
H2O: 1.5 mg/mL (3.03 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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AZ10606120 dihydrochloride 607378-18-7 Membrane transporter/Ion channel Neuroscience P2X Receptor AZ-10606120 dihydrochloride AZ 10606120 Inhibitor P2XRs AZ-10606120 Dihydrochloride inhibit AZ 10606120 Dihydrochloride AZ-10606120 AZ10606120 AZ10606120 Dihydrochloride inhibitor