Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study of cardiovascular and neurovascular diseases.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 78,500 |
5 mg | 在庫あり | ¥ 190,000 |
10 mg | 在庫あり | ¥ 264,000 |
25 mg | 在庫あり | ¥ 385,500 |
50 mg | 在庫あり | ¥ 525,500 |
100 mg | 在庫あり | ¥ 682,000 |
説明 | CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study of cardiovascular and neurovascular diseases. |
ターゲット&IC50 | CGRP receptor:35 nM(Ki), CGRP receptor:57 nM |
分子量 | 494.54 |
分子式 | C29H26N4O4 |
CAS No. | 1123757-49-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 60 mg/mL (121.32 mM)
You can also refer to dose conversion for different animals. 詳細
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CGRP antagonist 1 1123757-49-2 GPCR/G Protein Neuroscience CGRP Receptor Inhibitor inhibitor inhibit