Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ (pKis: 8.58, 8.49, and 8.71 for the human, rat, and mouse).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 28,000 | |||
5 mg | 在庫あり | ¥ 59,500 | |||
10 mg | 在庫あり | ¥ 100,500 | |||
25 mg | 在庫あり | ¥ 164,000 | |||
50 mg | 在庫あり | ¥ 226,000 | |||
100 mg | 在庫あり | ¥ 303,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 59,500 |
説明 | CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ (pKis: 8.58, 8.49, and 8.71 for the human, rat, and mouse). |
ターゲット&IC50 | Apelin receptor (human):pki:8.58 , Apelin receptor (rat):8.49 (pki), Apelin receptor (mouse):8.71(pki) |
分子量 | 455.61 |
分子式 | C25H33N3O3S |
CAS No. | 1586787-08-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 18.33 mg/mL (40.24 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
CMF019 1586787-08-7 GPCR/G Protein Apelin receptor CMF 019 CMF-019 Inhibitor inhibitor inhibit