store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Darbufelone mesylate (CI-1004 mesylate) inhibited PGF2α and LTB4 in cells. Darbufelone mesylate inhibited PGHS-2 with IC50 value of 0.19 μM and PGHS-1 with IC50 value of 20 μM.
パッケージサイズ | 在庫状況 | 単価(税別) | |
---|---|---|---|
5 mg | 在庫あり | ¥ 28,000 | |
10 mg | 在庫あり | ¥ 45,500 | |
25 mg | 約6-8 週間 | ¥ 104,500 | |
50 mg | 約6-8 週間 | お問い合わせ |
ターゲット&IC50 | PGHS1:20 μM, PGHS2:0.19 μM, H520:21μM, PGHS2:10±5 μM(Ki), A549 cells:20μM, PGHS2:0.98 ± 0.03μM(Kd) |
別名 | CI-1004 mesylate |
分子量 | 428.57 |
分子式 | C19H28N2O5S2 |
CAS No. | 139340-56-0 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (233.33 mM), Sonication is recommended.
H2O: <0.1mg/mL
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Darbufelone mesylate 139340-56-0 GPCR/G Protein Immunology/Inflammation LTR Prostaglandin Receptor CI 1004 Mesylate Darbufelone Mesylate CI1004 Mesylate CI-1004 Mesylate CI-1004 mesylate Inhibitor inhibitor inhibit