Powder: -20°C for 3 years | In solvent: -80°C for 1 year
ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 49,000 |
5 mg | 在庫あり | ¥ 123,500 |
10 mg | 在庫あり | ¥ 178,000 |
25 mg | 在庫あり | ¥ 273,500 |
50 mg | 在庫あり | ¥ 365,000 |
100 mg | 在庫あり | ¥ 498,000 |
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 136,000 |
説明 | ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively. |
ターゲット&IC50 | ERK2:3.0 nM, ERK1: |
In vitro | ERK1/2 inhibitor 1 ?shows excellent antiproliferative potency with IC50s of 7.5 and 4.9 nM in ?Colo205 cells and A375, respectively. |
分子量 | 550.05 |
分子式 | C29H32ClN5O4 |
CAS No. | 2095719-90-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 5.5 mg/mL (10 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
ERK1/2 inhibitor 1 2095719-90-5 MAPK ERK ERK-1/2 inhibitor 1 Inhibitor inhibitor inhibit