Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | お問い合わせ | |||
2 mg | 在庫あり | お問い合わせ | |||
5 mg | 在庫あり | お問い合わせ | |||
10 mg | 在庫あり | ¥ 238,500 | |||
25 mg | 在庫あり | ¥ 390,000 | |||
50 mg | 在庫あり | お問い合わせ | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 112,000 |
説明 | Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2. |
ターゲット&IC50 | ERRβ:0.66 nM(EC50) |
別名 | LY500307 |
分子量 | 282.33 |
分子式 | C18H18O3 |
CAS No. | 533884-09-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: 57 mg/mL (201.89 mM)
DMSO: 57 mg/mL (201.89 mM)
H2O: <1 mg/mL
You can also refer to dose conversion for different animals. 詳細
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Erteberel 533884-09-2 Endocrinology/Hormones Estrogen/progestogen Receptor Estrogen Receptor/ERR Inhibitor inhibit LY 500307 LY500307 LY-500307 inhibitor