Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD). CMP8 has IC50 values of 29 nM , 41 nM, 1100 nM and 2200 nM for MGERα, MGRERα, hERα and hERβ, respectively.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 58,000 |
5 mg | 在庫あり | ¥ 119,500 |
10 mg | 在庫あり | ¥ 170,500 |
25 mg | 在庫あり | ¥ 264,000 |
50 mg | 在庫あり | ¥ 356,000 |
100 mg | 在庫あり | ¥ 454,500 |
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 150,000 |
説明 | CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD). CMP8 has IC50 values of 29 nM , 41 nM, 1100 nM and 2200 nM for MGERα, MGRERα, hERα and hERβ, respectively. |
ターゲット&IC50 | MGRERα:41 nM, MGERα:29 nM, ERα (human):1100 nM, ERβ (human):2200 nM |
In vivo | CMP8 is dosed in male Balb-c mice (4 mg/kg, ip). In mammalian cells, the plasma concentration after 4 h is 1.5-fold its EC50. It has a Cmax of 0.5 μM after 30 min.[1][2] |
分子量 | 528.08 |
分子式 | C33H34ClNO3 |
CAS No. | 851107-28-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (94.68 mM)
You can also refer to dose conversion for different animals. 詳細
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CMP8 851107-28-3 Endocrinology/Hormones Estrogen Receptor/ERR Estrogen/progestogen Receptor inhibit CMP 8 Inhibitor CMP-8 inhibitor