Powder: -20°C for 3 years | In solvent: -80°C for 1 year
KDM2A/7A-IN-1 is a cell-permeable and selective inhibitor of the histone lysine demethylase KDM2A/7A with potential antitumor activity for the study of duodenal adenomas and ossifying fibromucoid tumors.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 62,500 |
5 mg | 在庫あり | ¥ 152,000 |
10 mg | 在庫あり | ¥ 243,500 |
25 mg | 在庫あり | ¥ 480,000 |
50 mg | 在庫あり | ¥ 638,000 |
100 mg | 在庫あり | ¥ 849,500 |
説明 | KDM2A/7A-IN-1 is a cell-permeable and selective inhibitor of the histone lysine demethylase KDM2A/7A with potential antitumor activity for the study of duodenal adenomas and ossifying fibromucoid tumors. |
ターゲット&IC50 | KDM2A:0.16 μM |
In vitro | KDM2A/7A-IN-1 is a highly cell-permeable inhibitor of KDM2A/7A, with an IC50 of 0.16 μM. KDM2A/7A-IN-1 (0.4, 3.1, 6.2 μM) increases the level of H3K36me2 in HeLa cells with ectopic expression of catalytically active KDM2A[1]. |
分子量 | 506.68 |
分子式 | C33H38N4O |
CAS No. | 2169272-46-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 120 mg/mL (236.84 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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KDM2A/7A-IN-1 2169272-46-0 Chromatin/Epigenetic Histone Demethylase KDM-2A/7A-IN-1 KDM2A/7AIN1 KDM2A/7A IN 1 Inhibitor inhibitor inhibit