Powder: -20°C for 3 years | In solvent: -80°C for 1 year
NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively)
説明 | NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively) |
ターゲット&IC50 | mGluR5:82 nM, mGluR1:5.2nM |
In vitro | Treatment of NPS2390 was conducive to inhibit the proliferation and reverse phenotypic modulation of PASMCs by regulating autophagy levels. |
分子量 | 307.39 |
分子式 | C19H21N3O |
CAS No. | 226878-01-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 3.07 mg/mL (10 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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NPS2390 226878-01-9 Neuroscience GluR Inhibitor Calcium-sensing receptor NPS 2390 mGluR inhibit Metabotropic glutamate receptors CaSR NPS-2390 inhibitor