Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 30,500 | |||
5 mg | 在庫あり | ¥ 69,500 | |||
10 mg | 在庫あり | ¥ 104,000 | |||
25 mg | 在庫あり | ¥ 171,500 | |||
50 mg | 在庫あり | ¥ 241,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 89,500 |
説明 | PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5. |
ターゲット&IC50 | Nav1.7 (human):21 nM (IC50) |
別名 | PF-05150122 |
分子量 | 531.89 |
分子式 | C19H10ClF4N5O3S2 |
CAS No. | 1235406-03-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 11 mg/mL (20.68 mM)
You can also refer to dose conversion for different animals. 詳細
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PF-05186462 1235406-03-7 Membrane transporter/Ion channel Sodium Channel acute Na channels PF05186462 inhibit chronic voltage PF-05150122 channel Na+ channels Inhibitor Nav1.7 pain PF 05150122 PF 05186462 sodium PF05150122 inhibitor