store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PKC-IN-1 is an ATP-competitive and reversible conventional PKC enzymes inhibitor (PKCα, PKCβI, PKCβII, PKCθ, PKCγ, PKC mu and PKCε with IC50s of 2.3, 8.1, 7.6, 25.6, 57.5, 314, 808 nM, respectively).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
2 mg | 在庫あり | ¥ 45,500 |
5 mg | 約8-10 週間 | ¥ 80,000 |
25 mg | 約8-10 週間 | ¥ 262,000 |
50 mg | 約8-10 週間 | ¥ 342,000 |
100 mg | 約8-10 週間 | ¥ 457,000 |
1 mL * 10 mM (in DMSO) | 約8-10 週間 | ¥ 88,000 |
ターゲット&IC50 | PKCγ (human):57.5 nM, PKCμ (human):314 nM, PKCε (human):808 nM, PKCβI (human):8.1 nM, PKCβ (human):5.3 nM (ki), PKCβII (human):7.6 nM, PKCθ (human):25.6 nM, PKCα (human):10.4 nM (ki), PKCα (human):2.3 nM |
分子量 | 500.61 |
分子式 | C25H37FN8O2 |
CAS No. | 1046787-18-1 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 25 mg/mL (49.94 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
PKC-IN-1 1046787-18-1 Chromatin/Epigenetic Cytoskeletal Signaling PKC PKCIN1 PKC IN 1 Protein kinase C inhibit Inhibitor inhibitor