Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ro 5212773 (Epptb) is a selective TAAR1 antagonist.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 7,500 | |||
5 mg | 在庫あり | ¥ 16,500 | |||
10 mg | 在庫あり | ¥ 29,500 | |||
25 mg | 在庫あり | ¥ 65,500 | |||
50 mg | 在庫あり | ¥ 131,000 | |||
100 mg | 在庫あり | ¥ 187,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 18,500 |
説明 | Ro 5212773 (Epptb) is a selective TAAR1 antagonist. |
ターゲット&IC50 | TAAR1:28 nM |
In vivo | EPPTB prevents the reduction of the firing frequency of DA neurons induced by p-tyramine (p-tyr), a nonselective TAAR1 agonist. the EPPTB effects were absent in Taar1 knockout mice, ruling out off-target effects[2]. |
別名 | Epptb |
分子量 | 378.39 |
分子式 | C20H21F3N2O2 |
CAS No. | 1110781-88-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/ml (145.35 mM)
You can also refer to dose conversion for different animals. 詳細
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Ro 5212773 1110781-88-8 Others Ro-5212773 Inhibitor Epptb neuronal inhibit Ro5212773 mesolimbic system TAAR1 GPCR inhibitor