Powder: -20°C for 3 years | In solvent: -80°C for 1 year
AChE/BChE-IN-10 is a potent dual inhibitor of AChE and BChE with IC50 values of 0.176, and 0.47 μM, respectively. AChE/BChE-IN-10 exhibits good blood brain barrier permeability. AChE/BChE-IN-10 can inhibit Aβ-aggregation.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
5 mg | 在庫あり | ¥ 16,000 | |||
10 mg | 在庫あり | ¥ 25,000 | |||
25 mg | 在庫あり | ¥ 52,500 | |||
50 mg | 在庫あり | ¥ 85,500 | |||
100 mg | 在庫あり | ¥ 124,000 | |||
500 mg | 在庫あり | ¥ 268,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 19,500 |
説明 | AChE/BChE-IN-10 is a potent dual inhibitor of AChE and BChE with IC50 values of 0.176, and 0.47 μM, respectively. AChE/BChE-IN-10 exhibits good blood brain barrier permeability. AChE/BChE-IN-10 can inhibit Aβ-aggregation. |
ターゲット&IC50 | AChE:0.176 μM, BChE:0.47 μM |
In vitro | AChE/BChE-IN-10 inhibits AChE in a non-competitive manner (Ki= 0.21 μM), and BChE in a mixed-fashion(Ki= 0.15 μM)[1]. |
分子量 | 402.53 |
分子式 | C26H30N2O2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 4.03 mg/mL (10 mM)
You can also refer to dose conversion for different animals. 詳細
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AChE/BChE-IN-10 Neuroscience AChR AChE Inhibitor inhibitor inhibit