store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Camonsertib (RP-3500) is a selective, orally active ATR kinase inhibitor (ATRi) with an IC50: 1.00 nM in biochemical assays and exhibits potent antitumour effects. Camonsertib is 30 times more selective for ATR than mTOR (IC50: 120 nM) and is a more active inhibitor of ATM, DNA-PK and PI3Kα kinases. PK and PI3Kα kinases.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 48,000 |
5 mg | 在庫あり | ¥ 121,500 |
10 mg | 在庫あり | ¥ 176,500 |
25 mg | 在庫あり | ¥ 273,500 |
50 mg | 在庫あり | ¥ 363,000 |
100 mg | 在庫あり | ¥ 496,000 |
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 136,000 |
説明 | Camonsertib (RP-3500) is a selective, orally active ATR kinase inhibitor (ATRi) with an IC50: 1.00 nM in biochemical assays and exhibits potent antitumour effects. Camonsertib is 30 times more selective for ATR than mTOR (IC50: 120 nM) and is a more active inhibitor of ATM, DNA-PK and PI3Kα kinases. PK and PI3Kα kinases. |
ターゲット&IC50 | ATR kinase:1 nM, mTOR:120 nM |
別名 | ATR inhibitor 4, RP-3500 |
分子量 | 410.47 |
分子式 | C21H26N6O3 |
CAS No. | 2417489-10-0 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45.0 mg/mL (109.6 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Camonsertib 2417489-10-0 DNA Damage/DNA Repair PI3K/Akt/mTOR signaling ATM/ATR ATR inhibitor 4 RP-3500 RP3500 RP 3500 Inhibitor inhibitor inhibit