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T1024 |
Roflumilast
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B9302-107,BYK 20869,APTA 2217,BY 217 |
PDE
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RSV
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Roflumilast (APTA 2217) is an orally available, long-acting inhibitor of phosphodiesterase (PDE) type 4 (PDE4), with anti-inflammatory and potential antineoplastic activities. Upon administration, roflumilast and its act... |
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T28167 |
NGB 2904
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NGB2904 HCl,NGB-2904,NGB2904 |
Others
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Dopamine Receptor
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5-HT Receptor
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NGB 2904 is a potent and selective antagonist of dopamine D3 receptor (Ki values are 1.4, 217, 223, 642, > 5000, > 10000 and > 10000 nM for D3, D2, 5-HT2, α1, D4, D1 and D5 receptors respectively). NGB2904 potently antag... |
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T37728 |
Methoctramine (hydrate)
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Methoctramine is a selective antagonist of M2 muscarinic acetylcholine receptors (IC50 = 6.1 nM in CHO-K1 cell membranes).[1] It is selective for M2 over M1, M3, M4, and M5 receptors (IC50s = 92, 770, 260, and 217 nM, re... |
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T36137 |
Biotin (S)-sulfoxide
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Biotin (S)-sulfoxide is an inactive metabolite of the coenzyme biotin .1,2It has also been found inE. coliand is reduced by the biotin sulfoxide reduction system as a source of biotin.3
1.Denkel, L.A., Rhen, M., and Bang... |
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T37018 |
OH-Chol
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OH-Chol is a cationic cholesterol derivative.1 OH-Chol, as a component of lipoplexes with DOPE , has been used for siRNA delivery and gene silencing in MCF-7 cells, as well as in mice via intravenous injection, resulting... |
