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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T3597 | Cutamesine dihydrochloride | AGY94806 dihydrochloride,SA4503 (dihydrochloride),SA4503 dihydrochloride | Sigma receptor |
Cutamesine dihydrochloride (SA4503 dihydrochloride) is a selective σ1 receptor agonist (IC50: 17.4 nM). It shows selectivity for σ1 over σ2 receptors, and inhibits angiotensin II-induced cardiomyocyte hypertrophy in vitr... |