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T82176 |
HR1
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HR1, a mastoid protease, enhances the permeability of human erythrocyte membranes and can induce cytoplasmic membrane permeation in bacteria and mast cells [1]. |
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T11966 |
MCHR1 antagonist 2
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HER
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Melanin-concentrating Hormone Receptor (MCHR)
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T68796 |
Thr101
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Others
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Thr101, also known as NOX Inhibitor VII, is a dose-dependent inhibitor of HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, and HDAC9. Thr101 is also a NOX inhibitor. |
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T10173 |
MCHR1 antagonist 1
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Others
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MCHR1 antagonist 1 is a selective antagonist of melanin-concentrating hormone-1 (MCH1) receptor (Kb: 1 nM, Ki: 4 nM at human MCH1). |
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T12904 |
SHR1653
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Others
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SHR1653 is a highly potent, selective and brain penetrated antagonist of oxytocin receptor (OTR)(IC50 of 15 nM for hOTR). |
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T39960 |
SHR168442
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SHR168442 |
Others
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SHR168442 is a potent RORγ modulator, exhibiting an IC50 value of 0.035 μM. |
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T11965 |
MCHR1 antagonist 3
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Others
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MCHR1 antagonist 3, a potent antagonist of the melanin-concentrating hormone receptor-1 (MCHR1), is employed for the regulation of energy metabolism. |
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T76270 |
SARS-CoV-2-IN-34
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SARS-CoV-2-IN-34 (S-20-1) is a broad-spectrum pan-coronavirus (CoV) fusion inhibitor capable of penetrating the blood-brain barrier and demonstrating extensive inhibitory activity against both pseudotyped and authentic S... |
