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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T2239L | Raltegravir | MK-0518 | HIV Protease , Integrase |
Raltegravir (MK-0518) is a pyrrolidinone derivative and HIV INTEGRASE INHIBITOR that is used in combination with other ANTI-HIV AGENTS for the treatment of HIV INFECTION. | |||
T2239 | Raltegravir potassium | MK 0518 potassium salt,Raltegravir potassium salt | HIV Protease , Integrase |
Raltegravir potassium (MK 0518 potassium salt) salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection. | |||
T62983 | Raltegravir sodium | ||
Raltegravir (MK 0518) sodium is a potent, orally active HIV integrase (IN) inhibitor. | |||
T2329 | Dolutegravir sodium | GSK1349572,GSK-1349572A | HIV Protease |
Dolutegravir sodium (GSK-1349572A) salt(DTG; GSK1349572) is an HIV integrase inhibitor(IC50: 2.7 nM), modest activity against raltegravir-resistant signature mutants Y143R, Q148K, N155H, and G140S/Q148H. | |||
T6198 | Dolutegravir | S/GSK1349572,GSK1349572 | HIV Protease |
Dolutegravir (GSK1349572) (IC50=2.7 nM), a two-metal-binding HIV integrase inhibitor, exhibits medium activity against raltegravir-resistant signature mutants Y143R, Q148K, N155H, and G140S/Q148H. | |||
T33443 | MK-8970 | ||
MK-8970 is an acetal carbonate prodrug of raltegravir with enhanced colonic absorption. |