4
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T6199 | Ribociclib | LEE011 | VEGFR , CDK |
Ribociclib (LEE011) is an orally available, and highly specific CDK4/6 inhibitor (IC50:10/39 nM). | |||
T15732 | Ribociclib succinate | LEE011 succinate | CDK |
Ribociclib succinate (LEE011 succinate) is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively). It also is over 1,000-fold less potent against the cyclin B/CDK1 complex. | |||
T15731 | Ribociclib succinate hydrate | LEE011 succinate hydrate | CDK |
T15730 | Ribociclib hydrochloride | LEE011 hydrochloride | CDK |