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T12939 |
SMYD2-IN-1
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|
Histone Methyltransferase
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SMYD2-IN-1 is an inhibitor of SMYD2 (IC50 of 4.45 nM). |
|
T6879 |
LLY-507
|
LLY507,LLY 507 |
Histone Methyltransferase
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|
LLY-507 is an effective, cell-active, and specific inhibitor of protein-lysine Methyltransferase SMYD2. |
|
TQ0100 |
AZ505
|
|
Histone Methyltransferase
|
|
AZ505 is an effective and specific SMYD2 inhibitor (IC50: 0.12 μM). |
|
T7403 |
BAY-598
|
|
Histone Methyltransferase
|
|
BAY-598 is a selective inhibitor of SMYD2 with IC50 values of 27 nM. |
|
T70087 |
EPZ032597
|
|
Histone Methyltransferase
|
|
EPZ032597 is a novel selective inhibitor of SMYD2 with an IC50 of 16 nM. EPZ032597 has anticancer activity and can be used to prevent and treat pancreatic cancer. |
|
T10427 |
AZ505 ditrifluoroacetate
|
|
Histone Methyltransferase
|
|
AZ505 ditrifluoroacetate is an effective and selective SMYD2 inhibitor (IC50: 0.12 μM). |
|
T5381 |
A-893
|
|
|
|
A-893 is a cell-active inhibitor of Methyltransferase SMYD2 (IC 50 = 2.8 nM) . |
|
T63783 |
AZ506
|
|
|
|
AZ506 is a potent inhibitor of SMYD2 (IC50: 17 nM). AZ506 inhibits SMYD2 methyltransferase activity in cells and reduces SMYD2-mediated methylation signaling. |
|
T26744 |
BAY-598 R-isomer
|
BAY598 R-isomer,BAY 598 R-isomer |
|
|
BAY-598 R-isomer is the R-isomer of BAY589, which is used as a reference compound. It is is an inhibitor of lysine N-methyltransferase (SMYD2) and is selective for SMYD2 over protease-activated receptor 1 (PAR1). |
