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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T2154 | MG-132 | Z-LLL-al,Z-Leu-Leu-Leu-CHO | Apoptosis , Proteasome , Autophagy |
MG-132 (Z-Leu-Leu-Leu-al) is a 26S proteasome inhibitor (IC50=100 nM) that is cell-permeable and reversible. MG-132 acts as an autophagy activator and also induces apoptosis. | |||
T78640 | Z-LLF-CHO | Z-Leu-Leu-Phe-CHO | Proteasome |
Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM. Additionally, this compound serves as an inhibitor of NF-κB ... | |||
T80735 | Z-Gly-Pro-Phe-Leu-CHO | Z-GPFL-CHO | Proteasome |
Z-Gly-Pro-Phe-Leu-CHO (Z-GPFL-CHO) is a tetrapeptide aldehyde serving as a selective and potent proteasome inhibitor, demonstrating inhibition constants (Ki) of 1.5 µM, 2.3 µM, and 40.5 µM for branched-chain amino acid-p... | |||
T17281 | Z-Ile-Leu-aldehyde | Z-IL-CHO,GSI-XII,γ-Secretase inhibitor XII | Others |
Z-Ile-Leu-aldehyde is an effective and competitive peptide aldehyde inhibitor of γ-secretase and notch. |