ペプチド
抗体
色素試薬
PROTAC
バーチャルスクリーニング
TargetMolキット
Cell Counting Kit-8 (CCK-8)
Inhibitor Cocktails
天然化合物
フェノール類
アルカロイド類
フラボノイド類
阻害剤
血管新生
アポトーシス
オートファジー
細胞周期・チェックポイント
クロマチン・エピジェネティック
細胞骨格シグナル
DNA損傷・DNA修復
内分泌・ホルモン
GPCR/Gタンパク質
免疫・炎症
JAK・STATシグナル
| Cat. No. | 製品名 | CAS No. | Purity | Chemical Structure |
|---|---|---|---|---|
| T16012 | Marizomib | 437742-34-2 | 98% |
|
| Marizomib is a novel irreversible brain-permeable proteasome inhibitor that inhibits CT-L (β5), CT-T-laspase-like (C-L, β1), and trypsin-like (T-L, β2) 20S prote... | ||||
| T2583 | Cilastatin | 82009-34-5 | 98% |
|
| Cilastatin is a renal dehydropeptidase-I and leukotriene D4 dipeptidase inhibitor. Since the antibiotic, IMIPENEM, is hydrolyzed by dehydropeptidase-I, which res... | ||||
| T7369L | Gemigliptin Tartrate(911637-19-9 free base) | 1374639-74-3 | 98% |
|
| Gemigliptin tartrate is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4). It has an IC50 of 10.3 nM for human recombina... | ||||
| T0242 | Sitagliptin | 486460-32-6 | 98% |
|
| Sitagliptin, a new oral hypoglycemic (anti-diabetic drug), is a new dipeptidyl peptidase-4 (DPP-4) inhibitor. This enzyme-inhibiting drug is used either alone or... | ||||
| T36902 | RA375 | 98% |
|
|
| RA375 is a inhibitor of RPN13 (26S proteasome regulatory subunit). RA375 activates UPR signaling, ROS production and apoptosis. RA375 exhibits ten-fold greater a... | ||||
| T2401 | Alogliptin Benzoate | 850649-62-6 | 98% |
|
| Alogliptin Benzoate(SYR 322), an effective and specific DPP-4 inhibitor (IC50<10 nM), exhibits greater than 10, 000-fold selectivity over DPP-8/9. Alogliptin may... | ||||
| T63321 | 20S Proteasome activator 1 | 2761578-18-9 | 98% |
|
| 20S Proteasome activator 1 is a 20S proteasome activator with IC50 of 0.3 μM for trypsin-like sites, 0.7 μM for chymotrypsin-like sites and 1.8 μM for caspase si... | ||||
| T16838 | Saikogenin A | 5092-09-1 | 98% |
|
| Saikogenin A is a dipeptidyl peptidase-4 inhibitor. | ||||
| T3359 | Aprotinin | 9087-70-1 | 98% |
|
| Aprotinin a broad-spectrum serine protease inhibitor, inhibiting the activity of a number of different esterases and proteases, including trypsin, chymotrypsin, ... | ||||
| T6203 | Saxagliptin | 361442-04-8 | 98% |
|
| Saxagliptin is a selective and reversible DPP4 inhibitor with IC50 of 26 nM. | ||||
| T2122 | Ixazomib | 1072833-77-2 | 98% |
|
| MLN2238, a second generation, boron-containing peptide proteasome inhibitor (PI), inhibits the chymotrypsin-like proteolytic (β5) site of the 20S proteasome (IC5... | ||||
| T7369 | Gemigliptin | 911637-19-9 | 98% |
|
| Gemigliptin is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.) | ||||
| T7814 | Alloxan monohydrate | 2244-11-3 | 98% |
|
| Alloxan Monohydrate is a glucose analog used to induce diabetes by destroying beta-cells. | ||||
| T2470 | MDL-28170 | 88191-84-8 | 98% |
|
| Calpain Inhibitor III is a Cysteine protease. | ||||
| T4042 | Talabostat mesylate | 150080-09-4 | 98% |
|
| Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation ... | ||||
| T7133 | Anagliptin | 739366-20-2 | 98% |
|
| Anagliptin is a potent Inhibitor of DPP-4(IC50 of 3.8 nM), for the treatment of type 2 diabetes mellitus. | ||||
| T6999 | Teneligliptin hydrobromide | 906093-29-6 | 98% |
|
| Teneligliptin is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-... | ||||
| T2296 | Trelagliptin succinate | 1029877-94-8 | 98% |
|
| Trelagliptin(SYR-472) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (T2D). | ||||
| T12079 | ML604440 | 1140517-08-3 | 98% |
|
| ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor. | ||||
| T2154 | MG-132 | 133407-82-6 | 98% |
|
| MG-132 is a potent cell-permeable 26S proteasome inhibitor (IC50: 100 nM). It also inhibits calpain (IC50: 1.2 μM). | ||||
