| T7369L |
Gemigliptin Tartrate(911637-19-9 free base)
|
1374639-74-3
|
98%
|
|
|
Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4). It has an IC50 of 10.3 n...
|
| T26754 |
BC-23
|
6298-15-3
|
98%
|
|
|
BC-23 (NSC 45382) is a potent proteasome inhibitor with antitumor and antimicrobial activity.BC-23 inhibits the CT-L activity of the proteasome and is used in th...
|
| T36902 |
RA375
|
|
98%
|
|
|
RA375, an inhibitor of RPN13 (26S proteasome regulatory subunit), enhances UPR signaling, ROS production, and apoptosis. Demonstrating ten times the efficacy aga...
|
| T3359 |
Aprotinin
|
9087-70-1
|
98%
|
|
|
Aprotinin (Traskolan) a broad-spectrum serine protease inhibitor, inhibiting the activity of a number of different esterases and proteases, including trypsin, ch...
|
| T7814 |
Alloxan monohydrate
|
2244-11-3
|
|
|
|
Alloxan Monohydrate is a glucose analog used to induce diabetes by destroying beta-cells.
|
| T2470 |
MDL-28170
|
88191-84-8
|
|
|
|
MDL-28170 (Calpain Inhibitor III) is a Cysteine protease.
|
| T6941 |
PI-1840
|
1401223-22-0
|
100%
|
|
|
PI-1840（IC50 = 27 nM）is a reversible and selective chymotrypsin-like (CT-L) inhibitor, with little proteasome proteolytic effects on trypsin-like (T-L) and postg...
|
| T7133 |
Anagliptin
|
739366-20-2
|
100%
|
|
|
Anagliptin (SK-0403) is a potent Inhibitor of DPP-4(IC50 of 3.8 nM), for the treatment of type 2 diabetes mellitus.
|
| T6999 |
Teneligliptin hydrobromide
|
906093-29-6
|
100%
|
|
|
Teneligliptin hydrobromide (MP-513 (hydrobromide)) is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, r...
|
| T2296 |
Trelagliptin succinate
|
1029877-94-8
|
100%
|
|
|
Trelagliptin succinate (SYR-472 succinate) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (T2...
|
| T12079 |
ML604440
|
1140517-08-3
|
95.24%
|
|
|
ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.
|
| T8350 |
TPCK
|
402-71-1
|
96.77%
|
|
|
TPCK is an irreversible inhibitor of chymotrypsin-like proteases that affect cell proliferation, apoptosis, and tumorigenesis
|
| T21617 |
MG-115
|
133407-86-0
|
97.12%
|
|
|
MG-115 (Z-LL-Nva-CHO) is a potent and reversible inhibitor of proteasome , with K i s of 21 nM and 35 nM for 20S and 26S proteasome, respectively. MG-115 specifi...
|
| T67852 |
Linagliptin Methyldimer
|
1418133-47-7
|
97.23%
|
|
|
Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.
|
| T16169 |
N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride
|
4272-74-6
|
97.44%
|
|
|
N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride (N-alpha-Tosyl-L-lysine_chloromethyl_ketone_hydrochloride) is an inhibitor of trypsin-like protease. N-a...
|
| T7854 |
Bortezomib-pinanediol
|
205393-22-2
|
97.5%
|
|
|
Bortezomib-pinanediol is a proteasome inhibitor. is a prodrug of Bortezomib.
|
| T6432 |
Calpeptin
|
117591-20-5
|
97.52%
|
|
|
Calpeptin is a potent, cell-permeable calpain inhibitor.
|
| T13858 |
RA190
|
1617495-03-0
|
97.69%
|
|
|
RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.
|
| TN1262 |
3-Feruloylquinic acid
|
1899-29-2
|
97.83%
|
|
|
3-O-Feruloylquinic acid is a protease inhibitor, it exerts moderate inhibitory effect against AIV (H5N1) in vitro.
|
| T7369 |
Gemigliptin
|
911637-19-9
|
98%
|
|
|
Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)
|
