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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T21534L | Oxytocin C-terminal tripeptide Acetate | Oxytocin C-terminal tripeptide Acetate(2002-44-0 Free base) | Others |
Oxytocin C-terminal tripeptide Acetate is the C-terminal tripeptide of Oxytocin.Oxytocin is a mammalian neuropituitary hormone, a ligand for the oxytocin receptor. | |||
T40536 | [Glu4]-Oxytocin | [Glu4]-Oxytocin | |
[Glu4]-Oxytocin is a suitable derivative of oxytocin for conducting a thorough investigation, utilizing various methods, into the conformation of "oxytocin-like" molecules in aqueous solution. | |||
T40534 | [Leu3]-Oxytocin | [Leu3]-Oxytocin | |
[Leu3]-Oxytocin, an oxytocin analogue, is a derivative of oxytocin wherein the leucine amino acid (Leu) has been substituted at the 3rd position in the sequence. | |||
T40756 | [Asp5]-Oxytocin | [Asp5]-Oxytocin | |
[Asp5]-Oxytocin is the first 5-position neurohypophyseal hormone analogue possessing significant biological activity. | |||
T40658 | [D-Asn5]-Oxytocin | [D-Asn5]-Oxytocin | |
[D-Asn5]-Oxytocin exhibits minimal specific oxytocic and vasodepressor effects. Comparative cumulative dose-response investigations reveal that [D-Asn5]-Oxytocin demonstrates a similar intrinsic activity to oxytocin in t... | |||
T33850 | Oxytocin, deamino-6-carba- | Deamino-6-carbaoxytocin,beta-Deaminocystathionine-oxytocin | |
Deamino-6-carba-oxytoxin (dC60), a potent oxytocin analog considered to be resistant to some of the physiologically significant enzymic systems. | |||
T40528 | Oxytocin free acid | 9-Deamidooxytocin | |
Oxytocin free acid, also known as 9-Deamidooxytocin, is an analog of oxytocin where the glycinamide residue at position 9 has been substituted with a glycine residue. Oxytocin, a pleiotropic peptide hormone, has wide-ran... | |||
T39388 | Oxytocin parallel dimer | ||
Oxytocin parallel dimer is the disulfide-bridged homo peptide dimer. | |||
T39420 | Oxytocin antiparallel dimer | ||
Oxytocin antiparallel dimer is the disulfide-bridged homo peptide dimer. | |||
T33849 | Oxytocin, deamino-1-carba- | Deamino-1-carbaoxytocin | |
Oxytocin, deamino-1-carba- is a biochemical. | |||
T80133 | Pro8-Oxytocin | Oxytocin Receptor | |
Pro8-Oxytocin, a modified oxytocin (OXT) ligand, elicits more potent and efficacious responses at primate OXTR and induces stronger behavioral effects compared to the standard mammalian OXT ligand (Leu8-Oxytocin). It dem... | |||
T76624 | (Ile8)-Oxytocin | ||
(Ile8)-Oxytocin is a neurohypophysial hormone mesotocin produced in marsupials [1] . | |||
T80136 | Val9-Oxytocin | Vasopressin Receptor | |
Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor. | |||
T80134 | Pro8-Oxytocin TFA | Oxytocin Receptor | |
Pro8-Oxytocin TFA, a modified oxytocin (OXT) ligand, exhibits greater potency and efficacy than the standard mammalian OXT ligand, Leu8-Oxytocin, at primate OXTR and elicits more pronounced behavioral effects. Compared t... | |||
T76629 | (Phe2,Orn8)-Oxytocin | ||
(Phe2,Orn8)-Oxytocin, a selective V1 vasopressin agonist, exhibits sustained contractility in rabbit epididymis, achieving an EC50 value of 280 nM [1]. | |||
T76265 | (Thr4,Gly7)-Oxytocin | ||
(Thr4,Gly7)-Oxytocin, an analogue of Oxytocin and a specific OT receptor agonist, not only activates TRPV1 channels to excite subicular neurons but also reduces the activity of potassium (K+) channels. [1] [2]. | |||
T80140 | (Val3,Pro8)-Oxytocin | Oxytocin Receptor | |
(Val3,Pro8)-Oxytocin functions primarily as a Gq-dependent pathway agonist and exhibits secondary activity as a reduced efficacy agonist for β-arrestin recruitment and receptor-mediated endocytosis at the oxytocin recept... | |||
T76211 | [Asp5]-Oxytocin acetate | ||
[Asp5]-Oxytocin acetate is a neurohypophyseal hormone analogue positioned at the 5-position, noted for its significant biological activity. It stimulates uterine contractions in vitro, an effect that is amplified by the ... | |||
T78021 | Oxytocin parallel dimer TFA | ||
Oxytocin Parallel Dimer TFA, a disulfide-bridged homopeptide dimer, exhibits both oxytocin and vasopressin-like activity while being less toxic than oxytocin [1] [2]. | |||
T76630 | (Phe2,Orn8)-Oxytocin acetate | ||
(Phe2,Orn8)-Oxytocin acetate, a selective V1 vasopressin agonist, demonstrates pronounced contractility induction in rabbit epididymis, characterized by a sustained response with an EC50 value of 280 nM [1]. | |||
T81583 | Oxytocin antiparallel dimer TFA | ||
Oxytocin antiparallel dimer TFA is a homo peptide dimer connected by a disulfide bridge, exhibiting activities similar to oxytocin and vasopressin but with reduced toxicity [1] [2]. | |||
T12331L | OT-R antagonist 1 | Oxytocin receptor antagonist 1 | Others |
OT-R antagonist 1 inhibits oxytocin-evoked intracellular Ca2+ mobilization (IC50 = 8 nM). OT-R antagonist 1 is a new effective and selective nonpeptide low molecular weight OT-R antagonist. | |||
T12331 | OT-R antagonist 2 | Oxytocin receptor antagonist 2 | Others |
OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R . | |||
T80126 | (d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin | Oxytocin Receptor | |
(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the study of neurological diseases [1]. | |||
T5148 | Atosiban acetate | RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164 | Oxytocin Receptor , Vasopressin Receptor |
Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban acetate (RW22164) inhibits... | |||
T11857 | LIT-001 | Oxytocin Receptor | |
LIT-001 improves social interaction in a mouse model of autism.It is the first nonpeptide oxytocin receptor agonist with EC50 of 55 nM and Ki of 226 nM. | |||
T4996 | Atosiban | RWJ22164,RW22164 | Oxytocin Receptor , Vasopressin Receptor |
Atosiban (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban inhibits the oxytocin-mediated rel... | |||
T7601L | Carbetocin acetate | Carbetocin acetate(37025-55-1 free base) | Oxytocin Receptor |
Carbetocin acetate is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth. | |||
T7601 | Carbetocin | Oxytocin Receptor | |
Carbetocin is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth. | |||
T76049 | Demoxytocin | ||
Demoxytocin, an analog of oxytocin and a heterodetic cyclic peptide, enhances cell membrane permeability to elevate calcium ion levels in smooth muscle cells, thereby augmenting contraction, including the smooth muscles ... | |||
T37694 | N-Acetyloxytocin | ||
N-Acetyloxytocin, a chemical compound, has been identified and analyzed in the neurointermediate lobe of the rat pituitary (NIL). Furthermore, its presence has also been detected in various brain regions of the rat[1]. | |||
T3347 | PF3274167 | PF 3274167,Cligosiban,PF-3274167 | OX Receptor |
PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist. | |||
T28855 | SSR126768A | SSR-126768A,SSR 126768A | Oxytocin Receptor |
SSR126768A is a novel and selective, orally active and potent oxytocin (OT) receptor antagonist with inhibitory effects on uterine contractions for the prevention of preterm labor. | |||
TP1400L | [Arg8]-Vasotocin acetate(113-80-4 free base) | Others | |
[Arg8]-Vasotocin acetate is a hormone present in the neurohypophysis of nonmammalian vertebrates that is related to vasopressin and oxytocin. | |||
T15682 | L-371,257 | Oxytocin Receptor , Vasopressin Receptor | |
L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a. | |||
TP2082L | D[Cha4]-AVP acetate(500170-27-4 free base) | Vasopressin Receptor | |
d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). Stimulates ACTH and corticosterone secre... | |||
T16736 | Retosiban | GSK 221149,GSK 221149A | Others |
Retosiban is an effective and selective oxytocin antagonist (Ki: 0.65 nM). | |||
T23528 | WAY-267464 | Others | |
oxytocin receptor (OTR) agonist | |||
T24278 | L 156373 | L-156373,L156373 | |
L 156373 is an oxytocin antagonist. | |||
T24288 | L 365209 | L365,209,L365209,L 365,209,L-365,209,L-365209 | |
L 365209 is an oxytocin antagonist. | |||
T69504 | Barusiban | ||
Barusiban is an oxytocin receptor antagonist. | |||
T23441 | TC OT 39 | Others | |
oxytocin receptor partial agonist | |||
T25902 | Ota-vasotocin | OVTA | |
Ota-vasotocin is a ligand utilized in quantitative receptor autoradiography for oxytocin receptors. | |||
T11502 | Epelsiban | GSK 557296 | Others |
T24291 | L 366811 | L 366,811,L-366,811,L366811,L366,811,L-366811 | |
L 366811 is a potent oxytocin antagonist. | |||
T27763 | L-366509 | L 366,509,L 366509,L366,509,L-366,509 | |
L-366,509 is an antagonist of oxytocin. | |||
T31647 | Epelsiban besylate | GSK-557296B,GSK557296B | |
Epelsiban Besylate is an oral drug that is a highly selective anamol oxytocin receptor antagonist. | |||
T12334 | OT antagonist 3 | Others | |
OT antagonist 3 is an antagonist of oxytocin (OT). | |||
T24289 | L 366682 | L366,682,L-66,682,L 366,682,L-366682,L366682 | |
L 366682 is an oxytocin antagonist. | |||
T24286 | L 364918 | L364,918,L-364918,L-364,918,L 364,918,L364918 | |
L 364918 is an oxytocin antagonist. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T5026 | Oxytocin | α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon) | Oxytocin Receptor |
Oxytocin (Oxytocin (Syntocinon)) is a mammalian neurohypophysial hormone, a ligand of oxytocin receptor. | |||
T5145 | Oxytocin acetate | Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base) | Oxytocin Receptor |
Oxytocin acetate (α-Hypophamine acetate) is a mammalian neurohypophysial hormone, a ligand of oxytocin receptor. | |||
T5065 | GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD | Monosodium-GMP,cGMP sodium salt,Cyclic GMP | PKA |
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD (cGMP sodium salt) , also known as cGMP, is a cellular regulatory agent and has been described as a second messenger. Its levels increase in response to a variety of hormones, inc... | |||
T36931 | Penicillide | ||
Penicillide is a fungal metabolite originally isolated from Penicillium that has diverse biological activities. It is an inhibitor of calpain 2/m-calpain (IC50 = 7.1 μM) and acyl-coenzyme A:cholesterol acyltransferase (A... |
カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPH-01820 | OXT Protein, Human, Recombinant (His) | Human | P. pastoris (Yeast) |
Neurophysin 1 specifically binds oxytocin.; Oxytocin causes contraction of the smooth muscle of the uterus and of the mammary gland. Acts by binding to oxytocin receptor (OXTR). OXT Protein, Human, Recombinant (His) is e... | |||
TMPH-01821 | OXT Protein, Human, Recombinant (His & Myc & SUMO) | Human | E. coli |
Neurophysin 1 specifically binds oxytocin.; Oxytocin causes contraction of the smooth muscle of the uterus and of the mammary gland. Acts by binding to oxytocin receptor (OXTR). OXT Protein, Human, Recombinant (His & Myc... | |||
TMPY-03269 | Prolyl Endopeptidase Protein, Mouse, Recombinant (His) | Mouse | Baculovirus Insect Cells |
Prolyl endopeptidase, also known as PREP, belongs to a distinct class of serine peptidases. It is a large cytosolic enzyme which was first described in the cytosol of rabbit brain as an oligopeptidase. Prolyl endopeptida... |