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カタログ番号 | 製品名 | 別名 | ターゲット |
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T10523 | β3-AR agonist 1 | Others | |
β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). | |||
T11804 | β3-AR agonist 2 | Others | |
β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM). | |||
T6872 | L755507 | Adrenergic Receptor , CRISPR/Cas9 | |
L755507 is an effective, selective agonist of β3-AR(IC50=35 nM). | |||
T12970 | Solabegron | GW 427353 | Adrenergic Receptor |
Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR(EC50 : 22 nM). It is used for treatment of overactive bladd... | |||
T34333 | Ritobegron HCl | KUC7483,KUC 7483,KUC-7483,Ritobegron,Ritobegron hydrochloride | |
Ritobegron (KUC-7483), an effective and selective β3-adrenergic receptor agonist, shows effective β(3)-AR agonist activity on transfected human β-AR and has an effect on the bladder of rats Shows high selectivity with ot... | |||
T63356 | Bopindolol fumarate | ||
Bopindolol ((±)-Bopindolol) fumarate is an orally active β-adrenoceptor (ARs) antagonist with partial agonist activity that is non-selective for β1- and β2-ARs and has low affinity for the β3-AR subtype. Bopindolol fumar... | |||
T2645 | Vilanterol | GW642444,GW642444X | Adrenergic Receptor |
Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma. | |||
T9451 | Bopindolol | ||
Bopindolol is an orally active antagonist of β-adrenoceptors (ARs) with partial agonist activity. Bopindolol is non-selective for β1- and β2-ARs and has low affinity for β3-AR subtype. Bopindolol is a prodrug of pindolol... |