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CaSR

The calcium-sensing receptor (CaSR) is a Class C G-protein coupled receptor which senses extracellular levels of calcium ion. It is primarily expressed in the parathyroid gland and the renal tubules of the kidney.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T29541 AC265347 1253901-26-6 98%
AC265347 is a potent calcium-sensitive receptor (CaSR) agonist and ago-PAM orthosteric modulator with antitumour activity that inhibits neuroblastoma tumour grow...
T40363 Poly-D-lysine hydrobromide (MW 30000-70000) 27964-99-4 98%
Poly-D-lysine hydrobromide (MW 30000-70000)(Poly-D-lysine HBr) is an orally available peptide CaSR agonist that removes proteinase K-resistant PrP from prion-inf...
T23401 Strontium chloride 10476-85-4 98%
Strontium chloride is an agonist of Calcium sensing receptor (CaSR) and directly affects C-type nerve fibers.
T12846 SB-423562 351490-27-2 98%
SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.
T22795 Gadolinium chloride 10138-52-0
Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
T1641 Strontium ranelate 135459-87-9 100%
Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis. Studies indicate it can also slow the course of osteoar...
TP1236 Etelcalcetide hydrochloride 1334237-71-6 100%
Etelcalcetide hydrochloride (AMG 416 hydrochloride) is a synthetic peptide as an allosteric modulator of the calcium (Ca)-sensing receptor (CaSR). Etelcalcetide ...
T1730 NPS-2143 284035-33-2 98.24%
NPS-2143 (SB 262470A) is a novel potent and selective antagonist of Ca(2+) receptor.
T29067L Upacicalcet HCl 98.56%
Upacicalcet HCl is an intravesical calcium mimetic that inhibits excessive parathyroid hormone (PTH) secretion by directly acting on calcium-sensitive receptors ...
T4967 NPS-2143 hydrochloride 324523-20-8 99.22%
NPS-2143 hydrochloride (NPS-2143 HCL) is a selective potent calcium ion-sensing receptor antagonist.
T13918 Tecalcet Hydrochloride 177172-49-5 99.44%
Tecalcet Hydrochloride (R-568 hydrochloride) is an allosteric and positive modulator of the calcium-sensing receptor(CaSR). Tecalcet Hydrochloride increases the ...
T3802 Ligustroflavone 260413-62-5 99.51%
Ligustroflavone (Nuezhenoside) has anti-inflammatory activity.
T34385 Ronacaleret HCl 702686-96-2 99.58%
Ronacaleret HCl (SB-751689) is a small molecule CaSR antagonist for the treatment of endocrine and metabolic diseases, skin and musculoskeletal disorders.
T8403 Cinacalcet 226256-56-0 99.82%
Cinacalcet (AMG 073) is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .
T15261 Evocalcet 870964-67-3 99.83%
Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).
T2406 Cinacalcet hydrochloride 364782-34-3 99.9%
Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-s...
T10666 Calhex 231 hydrochloride 2387505-78-2 98%
Calhex 231 hydrochloride is a CaSR inhibitor with the potential for diabetic cardiomyopathy treatment. It blocks Ca2+-induced accumulation of [3H]inositol phosph...
T79023 CaSR antagonist-1 1219811-83-2 98%
CaSR Antagonist-1 is a potent inhibitor of the calcium-sensing receptor (CaSR) with an inhibitory concentration (IC50) of 50 nM, suitable for the investigation o...
AC265347
T29541
AC265347 is a potent calcium-sensitive receptor (CaSR) agonist and ago-PAM orthosteric modulator with antitumour activity that inhibits neuroblastoma tumour grow...
Poly-D-lysine hydrobromide (MW 30000-70000)
T40363
Poly-D-lysine hydrobromide (MW 30000-70000)(Poly-D-lysine HBr) is an orally available peptide CaSR agonist that removes proteinase K-resistant PrP from prion-inf...
Strontium chloride
T23401
Strontium chloride is an agonist of Calcium sensing receptor (CaSR) and directly affects C-type nerve fibers.
SB-423562
T12846
SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.
Gadolinium chloride
T22795
Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
Strontium ranelate
T1641
Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis. Studies indicate it can also slow the course of osteoar...
Etelcalcetide hydrochloride
TP1236
Etelcalcetide hydrochloride (AMG 416 hydrochloride) is a synthetic peptide as an allosteric modulator of the calcium (Ca)-sensing receptor (CaSR). Etelcalcetide ...
NPS-2143
T1730
NPS-2143 (SB 262470A) is a novel potent and selective antagonist of Ca(2+) receptor.
Upacicalcet HCl
T29067L
Upacicalcet HCl is an intravesical calcium mimetic that inhibits excessive parathyroid hormone (PTH) secretion by directly acting on calcium-sensitive receptors ...
NPS-2143 hydrochloride
T4967
NPS-2143 hydrochloride (NPS-2143 HCL) is a selective potent calcium ion-sensing receptor antagonist.
Tecalcet Hydrochloride
T13918
Tecalcet Hydrochloride (R-568 hydrochloride) is an allosteric and positive modulator of the calcium-sensing receptor(CaSR). Tecalcet Hydrochloride increases the ...
Ligustroflavone
T3802
Ligustroflavone (Nuezhenoside) has anti-inflammatory activity.
Ronacaleret HCl
T34385
Ronacaleret HCl (SB-751689) is a small molecule CaSR antagonist for the treatment of endocrine and metabolic diseases, skin and musculoskeletal disorders.
Cinacalcet
T8403
Cinacalcet (AMG 073) is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .
Evocalcet
T15261
Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).
Cinacalcet hydrochloride
T2406
Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-s...
Calhex 231 hydrochloride
T10666
Calhex 231 hydrochloride is a CaSR inhibitor with the potential for diabetic cardiomyopathy treatment. It blocks Ca2+-induced accumulation of [3H]inositol phosph...
CaSR antagonist-1
T79023
CaSR Antagonist-1 is a potent inhibitor of the calcium-sensing receptor (CaSR) with an inhibitory concentration (IC50) of 50 nM, suitable for the investigation o...