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Glucocorticoid Receptor

The glucocorticoid receptor (GR, or GCR) also known as NR3C1 (nuclear receptor subfamily 3, group C, member 1) is the receptor to which cortisol and other glucocorticoids bind. The GR is expressed in almost every cell in the body and regulates genes controlling the development, metabolism, and immune response.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T0208 Prednisolone disodium phosphate 125-02-0
Prednisolone disodium phosphate, a synthetic glucocorticoid, has immunomodulating and anti-inflammatory properties.
T6022 LY404039 635318-11-5
LY404039 (pomaglumetad) is an effective agonist of recombinant human mGlu2(Ki =149 nM)/mGlu3(Ki =92 nM).
T6502 Fluocinonide 356-12-7 100%
Fluocinonide (Topsyn) (Vanos) is an effective glucocorticoid steroid, utilized in the treatment as the skin disorders anti-inflammatory agent.
T1683 Actriol 547-81-9 95.35%
Actriol (Epiestriol) is always used as Glucocorticoid Receptor agonist.
T2884 Cortisone 53-06-5 95.48%
Cortisone (17-Hydroxy-11-dehydrocorticosterone) is a corticosteroid with potent glucocorticoid activity.
T3096 Canrenoate potassium 2181-04-6 97.39%
Canrenoate potassium (Soldactone) is a synthetic pregnadiene derivative with anti-aldosterone activity.
T0947 Dexamethasone acetate 1177-87-3 98%
Dexamethasone acetate (NSC 39471) is the acetate salt form of Dexamethasone, a synthetic adrenal corticosteroid with potent anti-inflammatory properties. In addi...
T1749 AL 082D06 256925-03-8 98%
AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR(Ki > ...
T15000 Cort108297 1018679-79-2 98%
Cort108297 is a selective glucocorticoid receptor modulator and a selective GR antagonist with no affinity for other steroid receptors. Cort108297 showed a high ...
T15389L Glucagon (1-29), bovine, human, porcine hydrochloride 28270-04-4 98.03%
Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. It activates HNF4α and increases HNF4α phosphorylatio...
T1666 Fludrocortisone acetate 514-36-3 98.03%
Fludrocortisone acetate (9α-Fludrocortisone acetate) , a glucocorticoid-receptor agonist, binds to cytoplasmic receptors, translocates to the nucleus, and subseq...
T17217 Vamorolone 13209-41-1 98.04%
Vamorolone (VBP15) is an orally active dissociative steroidal anti-inflammatory drug and membrane-stabilizer. Vamorolone improves muscular dystrophy without side...
T6580 Meprednisone 1247-42-3 98.07%
Betapar(Meprednisone (Betapar)) is a glucocorticoid and a methylated derivative of prednisone.
T15102 Dexamethasone palmitate 14899-36-6 98.08%
Dexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone, shows a 47-fold lower affinity for the glucocorticoid receptor than Dexamethasone. Dexameth...
T2810 (20S)-Protopanaxatriol 34080-08-5 98.12%
(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid re...
T0294 6α-Methylprednisolone 21-hemisuccinate sodium salt 2375-03-3 98.16%
6α-Methylprednisolone 21-hemisuccinate sodium salt (Asmacortone), a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.
T3316 Fluorometholone 426-13-1 98.21%
Fluorometholone (Fluoromethalone) is a corticosteroid, most often used after laser-based refractive surgery. It is marketed under the brand names FML (Allergan) ...
T0034 Cortisone acetate 50-04-4 98.34%
Cortisone Acetate is a synthetic or semisynthetic analog of the naturally occurring cortisone hormone produced by the adrenal glands with anti-inflammatory and i...
T1561 Clobetasol propionate 25122-46-7 98.44%
Clobetasol propionate (CGP9555) exerts its effect by binding to cytoplasmic glucocorticoid receptors and subsequently activates glucocorticoid receptor-mediated ...
T4602 Hydrocortisone hemisuccinate 2203-97-6 98.7%
Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.
Prednisolone disodium phosphate
T0208
Prednisolone disodium phosphate, a synthetic glucocorticoid, has immunomodulating and anti-inflammatory properties.
LY404039
T6022
LY404039 (pomaglumetad) is an effective agonist of recombinant human mGlu2(Ki =149 nM)/mGlu3(Ki =92 nM).
Fluocinonide
T6502
Fluocinonide (Topsyn) (Vanos) is an effective glucocorticoid steroid, utilized in the treatment as the skin disorders anti-inflammatory agent.
Actriol
T1683
Actriol (Epiestriol) is always used as Glucocorticoid Receptor agonist.
Cortisone
T2884
Cortisone (17-Hydroxy-11-dehydrocorticosterone) is a corticosteroid with potent glucocorticoid activity.
Canrenoate potassium
T3096
Canrenoate potassium (Soldactone) is a synthetic pregnadiene derivative with anti-aldosterone activity.
Dexamethasone acetate
T0947
Dexamethasone acetate (NSC 39471) is the acetate salt form of Dexamethasone, a synthetic adrenal corticosteroid with potent anti-inflammatory properties. In addi...
AL 082D06
T1749
AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR(Ki > ...
Cort108297
T15000
Cort108297 is a selective glucocorticoid receptor modulator and a selective GR antagonist with no affinity for other steroid receptors. Cort108297 showed a high ...
Glucagon (1-29), bovine, human, porcine hydrochloride
T15389L
Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. It activates HNF4α and increases HNF4α phosphorylatio...
Fludrocortisone acetate
T1666
Fludrocortisone acetate (9α-Fludrocortisone acetate) , a glucocorticoid-receptor agonist, binds to cytoplasmic receptors, translocates to the nucleus, and subseq...
Vamorolone
T17217
Vamorolone (VBP15) is an orally active dissociative steroidal anti-inflammatory drug and membrane-stabilizer. Vamorolone improves muscular dystrophy without side...
Meprednisone
T6580
Betapar(Meprednisone (Betapar)) is a glucocorticoid and a methylated derivative of prednisone.
Dexamethasone palmitate
T15102
Dexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone, shows a 47-fold lower affinity for the glucocorticoid receptor than Dexamethasone. Dexameth...
(20S)-Protopanaxatriol
T2810
(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid re...
6α-Methylprednisolone 21-hemisuccinate sodium salt
T0294
6α-Methylprednisolone 21-hemisuccinate sodium salt (Asmacortone), a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.
Fluorometholone
T3316
Fluorometholone (Fluoromethalone) is a corticosteroid, most often used after laser-based refractive surgery. It is marketed under the brand names FML (Allergan) ...
Cortisone acetate
T0034
Cortisone Acetate is a synthetic or semisynthetic analog of the naturally occurring cortisone hormone produced by the adrenal glands with anti-inflammatory and i...
Clobetasol propionate
T1561
Clobetasol propionate (CGP9555) exerts its effect by binding to cytoplasmic glucocorticoid receptors and subsequently activates glucocorticoid receptor-mediated ...
Hydrocortisone hemisuccinate
T4602
Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.
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