Cat. No. | 製品名 | CAS No. | Purity | Chemical Structure |
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TP1819L | Substance P 1-9 aceate | 98% |
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Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder. | ||||
T77053 | Latozinemab | 98% |
Latozinemab
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Latozinemab (AL001) is a potent and selective recombinant humanized monoclonal antibody against Sortilin.Latozinemab has a high affinity for Sortilin and interru... | ||||
T38807L | [Lys8, Lys9]-Neurotensin (8-13) acetate | 98% |
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[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2, ... | ||||
TP1310 | Neurotensin | 39379-15-2 | 100% |
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Neurotensin is a 13 amino acid neuropeptide that is implicated in the regulation of luteinizing hormone and prolactin release and has significant interaction wit... | ||||
TP1116L | Kinetensin acetate(103131-69-7 free base) | TP1116L | 100% |
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Kinetensin acetate(103131-69-7 free base) is isolated from pepsin-treated human plasma. Kinetensin acetate(103131-69-7 free base) is a neurotensin-like peptide. | ||||
T7617L | Neurotensin(8-13) 3TFA(60482-95-3(free base)) | 2952825-79-3 | 100% |
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Neurotensin(8-13)(3TFA) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density. | ||||
T12848 | SB-657510 | 474960-44-6 | 98.03% |
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SB-657510 is a urotensin II (UII) receptor (UT) antagonist. The Ki values of UT for human, monkey, cat, rat and mouse were 61, 17, 30, 65 and 56 nM, respectively... | ||||
TP2106L | Urantide acetate(669089-53-6 free base) | TP2106L | 99.22% |
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Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. E... | ||||
T23323 | SB 611812 | 345892-71-9 | 99.34% |
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SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about the treatment of cardiovascular disease. | ||||
T22476 | (±)-AC 7954 hydrochloride | 477313-09-0 | 99.42% |
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(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator. | ||||
TQ0086 | AF38469 | 1531634-31-7 | 99.56% |
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AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM). | ||||
T9044 | SORT-PGRN interaction inhibitor 1 | 100957-85-5 | 99.56% |
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SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM). | ||||
T28217 | NTRC-844 | 1811503-67-9 | 99.61% |
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NTRC-844 is a selective rat neurotensin receptor type 2 (NTS2) antagonist that shows analgesic activity in animal models of pain. | ||||
T16860 | SBI-553 | 1849603-72-0 | 99.69% |
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SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM). | ||||
TP2104L | UFP 803 acetate | 99.78% |
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UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist. | ||||
TQ0075 | ML314 | 1448895-09-7 | 98% |
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ML314 is an effective molecule agonist of NTR1 (EC50: 1.9 μM). | ||||
T79106 | SORT-PGRN interaction inhibitor 3 | 2691846-87-2 | 98% |
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SORT-PGRN Interaction Inhibitor 3 (Compound 13), with an IC50 value of 0.17 μM, acts as an inhibitor of the SORT-PGRN interaction, and is utilized in the study o... | ||||
T79105 | BVFP | 357158-20-4 | 98% |
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BVFP exhibits affinity for the PGRN 588–593 peptide through binding with a dissociation constant (Kd) of 20 μM and is capable of disrupting the interaction betwe... | ||||
T78954 | HNTS1R agonist-1 | 98% |
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Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for hNTS1R (K i: 6.9 nM), showing the ability to cross the blood-brain barrier (B... | ||||
T23386 | SR 142948 | 184162-64-9 |
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SR 142948 is a neurotensin (NT) receptor antagonist. |