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Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T22850 ICI 204,448 121264-04-8 98%
ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.
TP2485 Difelikefalin acetate(1024828-77-0 Free base) TP2485 98%
is a ketone and a building block.
T21660L B-Casomorphin (1-3) Acetate T21660L 98%
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.
T12241 Norbinaltorphimine dihydrochloride 113158-34-2 98%
Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.
T13414 ZT 52656A hydrochloride 115730-24-0 98%
ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.
TP2036L DPDPE TFA (88373-73-3 free base) 172888-59-4 98%
DPDPE TFA is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is ant...
TP1832 Gluten Exorphin C 142479-62-7 98%
Gluten exorphin C is an opioid peptide derived from wheat gluten. Its IC50 values are 40 μM and 13.5 μM for μ opioid and δ opioid activities in the GPI and MVD a...
T5158 N-Desmethylclozapine 6104-71-8 98%
N-Desmethylclozapine (Desmethylclozapine) is an antagonist of serotonin (5-HT) receptor subtype 5-HT2C (IC50: 7.1 nM). It also is an antagonist at dopamine D4 re...
T7173 [Leu5]-Enkephalin 58822-25-6 98%
[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM,...
TP1211L BAM 22P acetate TP1211L 98%
BAM 22P acetate is a potent opioid agonist.
T20166 Deltorphin 119975-64-3 98%
Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.
TP1940L1 Ac-RYYRIK-NH2 acetate TP1940L1 98%
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial ag...
T4236 AR-M 1000390 hydrochloride 209808-47-9 98%
AR-M 1000390 hydrochloride (ARM-390 HCl) , also known as ARM-390, is a low-internalizing nonpeptidic δ-selective opioid receptor agonist; derivative of SNC 80. D...
T0201 Meptazinol hydrochloride 59263-76-2 98%
Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.
TP2052L CTOP acetate TP2052L 98%
CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.
TP1941L1 Ac-RYYRWK-NH2 acetate TP1941L1 98%
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.
T77445 Apitegromab 2278276-46-1 98%
Apitegromab
Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including spinal...
T14551 Bevenopran 676500-67-7 98%
Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.
T0918 Trimebutine 39133-31-8 98%
Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioid ag...
TP1826L Dynorphin B (1-13) acetate(83335-41-5 free base) TP1826L 98%
Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.
ICI 204,448
T22850
ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.
difelikefalin acetate(1024828-77-0 Free base)
TP2485
is a ketone and a building block.
b-Casomorphin (1-3) Acetate
T21660L
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.
Norbinaltorphimine dihydrochloride
T12241
Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.
ZT 52656A hydrochloride
T13414
ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.
DPDPE TFA (88373-73-3 free base)
TP2036L
DPDPE TFA is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is ant...
Gluten Exorphin C
TP1832
Gluten exorphin C is an opioid peptide derived from wheat gluten. Its IC50 values are 40 μM and 13.5 μM for μ opioid and δ opioid activities in the GPI and MVD a...
N-Desmethylclozapine
T5158
N-Desmethylclozapine (Desmethylclozapine) is an antagonist of serotonin (5-HT) receptor subtype 5-HT2C (IC50: 7.1 nM). It also is an antagonist at dopamine D4 re...
[Leu5]-Enkephalin
T7173
[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM,...
BAM 22P acetate
TP1211L
BAM 22P acetate is a potent opioid agonist.
Deltorphin
T20166
Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.
Ac-RYYRIK-NH2 acetate
TP1940L1
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial ag...
AR-M 1000390 hydrochloride
T4236
AR-M 1000390 hydrochloride (ARM-390 HCl) , also known as ARM-390, is a low-internalizing nonpeptidic δ-selective opioid receptor agonist; derivative of SNC 80. D...
Meptazinol hydrochloride
T0201
Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.
CTOP acetate
TP2052L
CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.
Ac-RYYRWK-NH2 acetate
TP1941L1
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.
Apitegromab
T77445
Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including spinal...
Bevenopran
T14551
Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.
Trimebutine
T0918
Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioid ag...
Dynorphin B (1-13) acetate(83335-41-5 free base)
TP1826L
Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.
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