keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial agonist on ORL1 transfected in CHO cells, antagonizes the stimulation of [35S]-GTPgammaS binding to G proteins by noc/OFQ in membranes and sections of rat brain.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 68,000 |
2 mg | 在庫あり | ¥ 102,000 |
5 mg | 在庫あり | ¥ 153,000 |
10 mg | 在庫あり | ¥ 229,000 |
25 mg | 在庫あり | ¥ 340,000 |
50 mg | 在庫あり | ¥ 457,000 |
100 mg | 在庫あり | ¥ 617,500 |
説明 | Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial agonist on ORL1 transfected in CHO cells, antagonizes the stimulation of [35S]-GTPgammaS binding to G proteins by noc/OFQ in membranes and sections of rat brain. |
In vivo | When administered intracerebroventricularly (i.c.v.), Ac-RYYRIK-NH inhibited spontaneous locomotor activity in mice with ID50 of 0.07 nmol, respectively[1]. |
分子量 | 999.17 |
分子式 | C46H74N14O11 |
CAS No. | TP1940L1 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Ac-RYYRIK-NH2 acetate TP1940L1 Endocrinology/Hormones GPCR/G Protein Neuroscience Opioid Receptor Ac-RYYRIK-NH2 Acetate Ac-RYYRIK-NH-2 acetate AcRYYRIKNH2 acetate Ac RYYRIK NH2 acetate Inhibitor inhibitor inhibit