ペプチド
抗体
色素試薬
PROTAC
バーチャルスクリーニング
TargetMolキット
Cell Counting Kit-8 (CCK-8)
Inhibitor Cocktails
天然化合物
フェノール類
アルカロイド類
フラボノイド類
阻害剤
血管新生
アポトーシス
オートファジー
細胞周期・チェックポイント
クロマチン・エピジェネティック
細胞骨格シグナル
DNA損傷・DNA修復
内分泌・ホルモン
GPCR/Gタンパク質
免疫・炎症
JAK・STATシグナル
| Cat. No. | 製品名 | CAS No. | Purity | Chemical Structure |
|---|---|---|---|---|
| T9256 | N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine | 1071135-06-2 | 98% |
|
| N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine is a novel 2,6-naphthyridine identified by high throughput screen (HTS) as a dual protein... | ||||
| TN3694 | Coniferaldehyde | 20649-42-7 | 98% |
|
| Coniferaldehyde can significantly inhibit the growth of viability of strains of Oenococcus oeni. Coniferaldehyde exerts anti-inflammatory properties by inducing ... | ||||
| T14072 | A-443654 | 552325-16-3 | 98% |
|
| A-443654 is a pan-Akt inhibitor. It has equal potency against Akt1, Akt2, or Akt3 within cells (Ki=160 pM). | ||||
| T7790 | Bisindolylmaleimide V | 113963-68-1 | 98% |
|
| Bisindolylmaleimide V (BIM V) is a weak protein kinase C (PKC)inhibitor( IC50 >100 µM) | ||||
| T6605 | NH125 | 278603-08-0 | 98% |
|
| NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, >125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor. | ||||
| T77628 | Bisindolylmaleimide III | 137592-43-9 | 98% |
|
| Bisindolylmaleimide III is a potent and selective inhibitor of protein kinase C (PKC).Bisindolylmaleimide III selectively interacts with PKCα or ribosomal S6 pro... | ||||
| T3211 | Midostaurin | 120685-11-2 | 98% |
|
| PKC412(Midostaurin; CGP41231; CGP41251) is a broad spectrum protein kinase inhibitor. Midostaurin inhibits protein kinase C alpha (PKCalpha), vascular endothelia... | ||||
| T13363 | Y06137 | 2226534-49-0 | 98% |
|
| Y06137 is an effective and selective BET inhibitor with a Kd of 81 nM for BRD4(1) bromodomain. Y06137 can be used for research on the treatment of castration-res... | ||||
| TP1888L1 | [Ala113]-MBP (104-118) acetate | TP1888L1 | 98% |
|
| [Ala113]MBP(104-118) acetate is an noncompetitive peptide inhibitors of protein kinase C (PKC), with IC50s ranging from 28-62 μM. | ||||
| T11665 | Ionomycin calcium | 56092-82-1 | 98% |
|
| lonomycin calcium is a potent, selective calcium ionophore and an antibiotic produced by Streptomyces conglobatus. also induces the activation of protein kinase ... | ||||
| T4444 | A-674563 HCl (552325-73-2(free base)) | 98% |
|
|
| A-674563 is an orally available, ATP-competitive, and reversible inhibitor of Akt (Ki: 11 nM for Akt1) [1]. It exhibits inhibitory activity against PKA and Cdk2 ... | ||||
| TP1887L1 | [Ala107]-MBP (104-118) acetate | TP1887L1 | 98% |
|
| [Ala107]-MBP (104-118) acetate is synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 46 - 145 mM). | ||||
| T60109 | Protein kinase inhibitor H-7 | 84477-87-2 | 98% |
|
| Protein kinase inhibitor H-7 is a potent inhibitor of protein kinase C (PKC) with a Ki of 6 μM. Protein kinase inhibitor H-7 is also a cyclic nucleotide dependen... | ||||
| T17019 | TCS 21311 | 1260181-14-3 | 98% |
|
| TCS 21311 is an effective and highly selective inhibitor of JAK3 (IC50: 8 nM). TCS 21311 inhibits PKCα, PKCθ, and GSK3β (IC50s: 13, 68, and 3 nM, respectively).... | ||||
| T22464 | 1,2-Dimyristoyl-sn-glycerol | 60562-16-5 | 98% |
|
| 1,2-dimyristoyl-sn-glycerol is able to increase AChE activity by 35-40% at concentrations of 25 micrograms/ml in the parasite S. mansoni.. | ||||
| T72322 | R 59-022 hydrochloride | 93076-98-3 | 98% |
|
| R 59-022 hydrochloride is a 5-HT Receptor antagonist that activates protein kinase C (PKC).R 59-022 hydrochloride is a DGK inhibitor (IC50:2.8 µM) that inhibits ... | ||||
| T35407 | Ζ-Stat | 3316-02-7 | 98% |
|
| ζ-Stat (NSC37044) is a specific and atypical PKC-ζ inhibitor, with an IC50 of 5 μM. ζ-Stat can reduce melanoma cell lines proliferation and induce apoptosis, and... | ||||
| T14943 | CGP60474 | 164658-13-3 | 98% |
|
| CGP60474 is an inhibitor of VEGFR-2 (IC50: 84 nM) and an ATP-competitive inhibitor of PKC. | ||||
| T6588 | Mitoxantrone | 65271-80-9 | 98% |
|
| Mitoxantrone is an anthracenedione antibiotic with antineoplastic activity. Mitoxantrone intercalates into and crosslinks DNA, thereby disrupting DNA and RNA rep... | ||||
| T5817 | PKC-theta inhibitor hcl | 2253640-49-0 | 98% |
|
| PKC-theta inhibitor is a selective PKC-θinhibitor(IC50:12 nM). | ||||
