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Protease-activated Receptor

Protease-activated receptors (PAR) are a subfamily of related G protein-coupled receptors that are activated by cleavage of part of their extracellular domain. They are highly expressed in platelets, and also on endothelial cells, myocytes and neurons.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T7513 Protease-Activated Receptor-2, amide 190383-13-2 98%
Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)
T7625 TRAP-6 141136-83-6 98%
TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).
T1893 Parmodulin 2 423735-93-7 98%
Parmodulin 2 (ML 161) is the inhibitor of protease-activated receptor 1 (PAR1)-mediated platelet activation (IC50: 0.26 μM for the inhibition of platelet P-selec...
T7674 Thrombin Receptor Activator for Peptide T7674 98%
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
TN6872 Trypsin 9002-07-7 98%
Trypsin is a serine protease that can be isolated from fish to hydrolyze lysine or arginine carboxy-side proteins. With the anti-inflammatory activity, Trypsin c...
T27267 ENMD-1068 HCl 789488-77-3 98%
ENMD-1068 HCl (ENMD 1068) is a PAR-2 antagonist. ENMD-1068 HCl inhibits the development of endometriosis in a mouse model.
T22933L LRGILS-NH2 acetate 98%
LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.
TP1904L FSLLRY-NH2 TFA(245329-02-6 free base) TP1904L
FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR...
T7623 PAR-4 Agonist Peptide, amide 352017-71-1
PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).
TP1065 PAR-4 Agonist Peptide, amide TFA 1228078-65-6 100%
PAR-4 Agonist Peptide, amide TFA (PAR-4-AP (TFA)) is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose ef...
TP1925L TcY-NH2 TFA(327177-34-4 free base) TP1925L 100%
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.
TP1378 2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) TP1378 100%
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.
T7573L TFLLR-NH2 2TFA(197794-83-5(free base)) T7573L 100%
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
T1986L Atopaxar Hydrobromide 474550-69-1 100%
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
T7137 I-191 1690172-25-8 98%
I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.
T38836L Protease-Activated Receptor-1, PAR-1 Agonist acetate 98.18%
Protease-Activated Receptor-1, PAR-1 Agonist acetate is a selective proteinase-activated receptor1 (PAR-1) agonist peptide. Protease-Activated Receptor-1, PAR-1 ...
T1986 Atopaxar 751475-53-3 98.25%
Atopaxar (E5555), a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Corona...
TQ0012 AZ3451 2100284-59-9 98.44%
AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
TP1046L PAR-2 Activating Peptide acetate TP1046L 98.5%
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).
T38852L TRAP-6 amide acetate 98.55%
TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].
Protease-Activated Receptor-2, amide
T7513
Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)
TRAP-6
T7625
TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).
Parmodulin 2
T1893
Parmodulin 2 (ML 161) is the inhibitor of protease-activated receptor 1 (PAR1)-mediated platelet activation (IC50: 0.26 μM for the inhibition of platelet P-selec...
Thrombin Receptor Activator for Peptide
T7674
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
Trypsin
TN6872
Trypsin is a serine protease that can be isolated from fish to hydrolyze lysine or arginine carboxy-side proteins. With the anti-inflammatory activity, Trypsin c...
ENMD-1068 HCl
T27267
ENMD-1068 HCl (ENMD 1068) is a PAR-2 antagonist. ENMD-1068 HCl inhibits the development of endometriosis in a mouse model.
LRGILS-NH2 acetate
T22933L
LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.
FSLLRY-NH2 TFA(245329-02-6 free base)
TP1904L
FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR...
PAR-4 Agonist Peptide, amide
T7623
PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).
PAR-4 Agonist Peptide, amide TFA
TP1065
PAR-4 Agonist Peptide, amide TFA (PAR-4-AP (TFA)) is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose ef...
tcY-NH2 TFA(327177-34-4 free base)
TP1925L
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
TP1378
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.
TFLLR-NH2 2TFA(197794-83-5(free base))
T7573L
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
Atopaxar Hydrobromide
T1986L
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
I-191
T7137
I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.
Protease-Activated Receptor-1, PAR-1 Agonist acetate
T38836L
Protease-Activated Receptor-1, PAR-1 Agonist acetate is a selective proteinase-activated receptor1 (PAR-1) agonist peptide. Protease-Activated Receptor-1, PAR-1 ...
Atopaxar
T1986
Atopaxar (E5555), a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Corona...
AZ3451
TQ0012
AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
PAR-2 Activating Peptide acetate
TP1046L
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).
TRAP-6 amide acetate
T38852L
TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].
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