Powder: -20°C for 3 years | In solvent: -80°C for 1 year
α-Glucosidase-IN-23 is an orally active α-Glucosidase inhibitor. α-Glucosidase-IN-23 can decrease blood glucose by α-glucosidase inhibition (IC50= 4.48 μM).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 75,500 |
5 mg | 在庫あり | ¥ 183,500 |
10 mg | 在庫あり | ¥ 250,500 |
25 mg | 在庫あり | ¥ 379,000 |
50 mg | 在庫あり | ¥ 512,000 |
100 mg | 在庫あり | ¥ 672,500 |
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 219,000 |
説明 | α-Glucosidase-IN-23 is an orally active α-Glucosidase inhibitor. α-Glucosidase-IN-23 can decrease blood glucose by α-glucosidase inhibition (IC50= 4.48 μM). |
In vitro | α-Glucosidase-IN-23 (1 μM) exhibits significant anti-diabetes activity. α-Glucosidase-IN-23 decreases ROS levles in βcells and muscle cells. α-Glucosidase-IN-23 decreases blood glucose by α-glucosidase inhibition (IC50= 4.48 μM)[1]. |
In vivo | α- Glucosidase-IN-23 (oral; 0.2 mmol/kg/day) only inhibits α- Glucosidase in mice[1]. |
分子量 | 373.4 |
分子式 | C20H23NO6 |
CAS No. | 161187-57-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 25 mg/mL (66.95 mM)
You can also refer to dose conversion for different animals. 詳細
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α-Glucosidase-IN-23 161187-57-1 Metabolism Glucosidase alpha-Glucosidase-IN-23 a-Glucosidase-IN-23 αGlucosidaseIN23 Inhibitor inhibitor inhibit