keep away from direct sunlight,store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
AZD9567 is a potent and orally active and selective non-steroidal glucocorticoid receptor modulator (SGRM) with an IC50 value of 3.8 nM.It has demonstrated excellent efficacy in the Streptococcus cell wall (SCW) reactivation model of joint inflammation.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 49,000 |
5 mg | 在庫あり | ¥ 123,500 |
10 mg | 在庫あり | ¥ 178,500 |
25 mg | 在庫あり | ¥ 271,000 |
50 mg | 在庫あり | ¥ 365,000 |
100 mg | 在庫あり | ¥ 489,000 |
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 136,000 |
説明 | AZD9567 is a potent and orally active and selective non-steroidal glucocorticoid receptor modulator (SGRM) with an IC50 value of 3.8 nM.It has demonstrated excellent efficacy in the Streptococcus cell wall (SCW) reactivation model of joint inflammation. |
ターゲット&IC50 | GR:3.8 nM |
In vivo | AZD9567 (15 mg/kg/day; Oral gavage; daily for 8 days; female Lewis rats; sensitized by intra-articular injection of 5 μg of SCW) inhibited ankle swelling in the rat SCW model. The treatment shows excellent in vivo efficacy in a rat model of joint inflammation.[1] |
別名 | Mizacorat |
分子量 | 494.53 |
分子式 | C27H28F2N4O3 |
CAS No. | 1893415-00-3 |
keep away from direct sunlight,store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (101.11 mM)
You can also refer to dose conversion for different animals. 詳細
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AZD9567 1893415-00-3 Endocrinology/Hormones Glucocorticoid Receptor Mizacorat AZD-9567 AZD 9567 Inhibitor inhibitor inhibit