Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Almorexant hydrochloride (ACT-078573 hydrochloride) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
2 mg | 約5 days | ¥ 16,000 |
5 mg | 約5 days | ¥ 27,500 |
10 mg | 約5 days | ¥ 47,000 |
25 mg | 約5 days | ¥ 94,000 |
50 mg | 約5 days | ¥ 165,000 |
100 mg | 約5 days | ¥ 267,000 |
1 mL * 10 mM (in DMSO) | 約5 days | ¥ 35,500 |
説明 | Almorexant hydrochloride (ACT-078573 hydrochloride) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively. |
ターゲット&IC50 | OX2:0.17 nM(ki), OX1:1.3 nM(ki) |
別名 | ACT-078573 hydrochloride, Almorexant HCl |
分子量 | 549.02 |
分子式 | C29H32ClF3N2O3 |
CAS No. | 913358-93-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: 48 mg/mL (87.4 mM)
DMSO: 67 mg/mL (122 mM)
H2O: <1 mg/mL
You can also refer to dose conversion for different animals. 詳細
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