Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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5 mg | 在庫あり | ¥ 13,000 | |||
10 mg | 在庫あり | ¥ 18,500 | |||
25 mg | 在庫あり | ¥ 30,000 | |||
50 mg | 在庫あり | ¥ 43,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 15,500 |
説明 | Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay). |
ターゲット&IC50 | Ghrelin receptor:(EC50)0.74 nM , Ghrelin receptor:(ki)0.7 nM |
In vitro | Anamorelin(ANAM) is a potent and highly specific ghrelin receptor agonist |
In vivo | Anamorelin(ANAM) showed significant agonist and binding activity on the ghrelin receptor, and stimulated GH release in vitro.?In rats, ANAM significantly and dose-dependently increased FI and BW at all dose levels compared with control, and significantly increased GH levels at 10 or 30 mg/kg doses.?Increases in GH and IGF-1 levels were observed following ANAM administration in pigs. |
別名 | RC-1291, ONO-7643 |
分子量 | 546.7 |
分子式 | C31H42N6O3 |
CAS No. | 249921-19-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (91.46 mM)
You can also refer to dose conversion for different animals. 詳細
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Anamorelin 249921-19-5 GPCR/G Protein GHSR Growth hormone secretagogue receptor RC-1291 Inhibitor RC 1291 ONO7643 ONO 7643 ONO-7643 RC1291 inhibit inhibitor