Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Calmidazolium chloride (R 24571) is a calmodulin (CaMK) antagonist (Kd = 3 nM), antagonizing CaM-dependent phosphodiesterase(IC50 = 0.15 μM) and calmodulin-induced activation of erythrocyte Ca2+-transporting ATPase(IC50 = 0.35 μM). Calmidazolium chloride also induces apoptosis in certain cancer cell lines.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
5 mg | 在庫あり | ¥ 13,000 | |||
10 mg | 在庫あり | ¥ 20,500 | |||
25 mg | 在庫あり | ¥ 34,000 | |||
50 mg | 在庫あり | ¥ 52,000 | |||
100 mg | 在庫あり | ¥ 77,500 | |||
200 mg | 在庫あり | ¥ 113,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 20,000 |
ターゲット&IC50 | PDE (CaM-dependent):0.15 μM, Calmodulin:12.69 μM(mouse E14 ESCs), Calmodulin:3 nM(kd), Calmodulin:8.18 μM(mouse F9 ECCs), Ca2+ transporting ATPase (erythrocyte, Calmodulin-induced):0.35 μM |
別名 | R 24571 |
分子量 | 687.7 |
分子式 | C31H23Cl7N2O |
CAS No. | 57265-65-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (145.41 mM)
You can also refer to dose conversion for different animals. 詳細
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Calmidazolium chloride 57265-65-3 Autophagy Neuroscience CaMK R-24571 Calmidazolium Inhibitor inhibit R 24571 Calmodulin-dependent protein kinases Calmodulin-dependent kinases R24571 Calmidazolium Chloride inhibitor