Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Cyclapolin 9 is a selective, potent, and ATP-competitive inhibitor of polo-like kinase 1 (PLK1) with an IC50 of 500 nM, and has not shown activity against other kinases.
説明 | Cyclapolin 9 is a selective, potent, and ATP-competitive inhibitor of polo-like kinase 1 (PLK1) with an IC50 of 500 nM, and has not shown activity against other kinases. |
ターゲット&IC50 | PLK1:500 nM |
In vitro | Reducing electric field stimulation (EFS)-induced contractions of prostate strips, Cyclapolin 9 (3 μM) has the ability to inhibit α1-adrenergic smooth muscle contraction in the human prostate[1] |
分子量 | 307.21 |
分子式 | C9H4F3N3O4S |
CAS No. | 40533-25-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: < 1 mg/mL (insoluble or slightly soluble)
DMSO: 10 mg/mL (32.55 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Cyclapolin 9 40533-25-3 Cell Cycle/Checkpoint PLK Inhibitor inhibitor inhibit