Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor (IC50: 47 nM).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 27,000 | |||
5 mg | 在庫あり | ¥ 108,000 | |||
10 mg | 在庫あり | ¥ 157,000 | |||
25 mg | 在庫あり | ¥ 226,500 | |||
50 mg | 在庫あり | ¥ 319,000 | |||
100 mg | 在庫あり | ¥ 431,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 102,500 |
説明 | DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor (IC50: 47 nM). |
ターゲット&IC50 | LTA4H:47 nM (IC50) |
In vitro | DG051 is a potent inhibitor of LTA4H aminopeptidase activity against L-alanine p-nitroanilide (IC50: 72 nM). DG051 inhibits human whole blood (HWB) with IC50 of 37 nM [1]. DG-051 is an LTA4H inhibitor, currently in Phase II clinical development for the prevention of heart attack [2]. |
分子量 | 426.33 |
分子式 | C21H25Cl2NO4 |
CAS No. | 929915-58-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 317 mg/mL (743.56 mM)
You can also refer to dose conversion for different animals. 詳細
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DG051 929915-58-2 Metabolism Aminopeptidase inhibit Inhibitor DG 051 DG-051 inhibitor