Powder: -20°C for 3 years | In solvent: -80°C for 1 year
ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substrates but competitively inhibits its activity toward a nonamer peptide representative of physiological substrates.
説明 | ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substrates but competitively inhibits its activity toward a nonamer peptide representative of physiological substrates. |
In vitro | ERAP1-IN-1 (50 μM) exhibits specific inhibition of ERAP1 in the cellular context. ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substrates. |
分子量 | 458.45 |
分子式 | C20H21F3N2O5S |
CAS No. | 865273-97-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL (545.32 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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ERAP1-IN-1 865273-97-8 Others ERAP1 IN 1 ERAP1 inhibit ERAP-1-IN-1 Inhibitor aminopeptidase ERAP1IN1 reticulum endoplasmic inhibitor