Powder: -20°C for 3 years | In solvent: -80°C for 1 year
L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 13,000 | |||
5 mg | 在庫あり | ¥ 32,000 | |||
10 mg | 在庫あり | ¥ 51,000 | |||
25 mg | 在庫あり | ¥ 102,500 | |||
50 mg | 在庫あり | ¥ 151,500 | |||
100 mg | 在庫あり | ¥ 215,500 |
説明 | L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a. |
ターゲット&IC50 | OTR:(ki)19 nM, V1a receptor:3.7 nM(ki) |
In vivo | L-371,257 (0.5 and 1.0 mg/kg; i.p.) stimulates weight gain (10.5 g) relative to vehicle treatment (4.7 g) in rats[3]. |
分子量 | 507.58 |
分子式 | C28H33N3O6 |
CAS No. | 162042-44-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 8.1 mg/mL (16 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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L-371,257 162042-44-6 Endocrinology/Hormones GPCR/G Protein Oxytocin Receptor Vasopressin Receptor L371,257 L 371,257 Inhibitor inhibitor inhibit