Powder: -20°C for 3 years | In solvent: -80°C for 1 year
ML254 competitively interacts with the MPEP allosteric binding site. ML254 is highly selective for mGlu5 versus other mGlu receptors, has a clean ancillary Ricerca profile, and suitable dystrophia myotonica protein kinase (DMPK) properties for systemic dosing in rodents.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 12,000 | |||
5 mg | 在庫あり | ¥ 28,000 | |||
10 mg | 在庫あり | ¥ 45,500 | |||
25 mg | 在庫あり | ¥ 104,500 | |||
50 mg | 在庫あり | ¥ 154,500 | |||
100 mg | 在庫あり | ¥ 219,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 36,000 |
説明 | ML254 competitively interacts with the MPEP allosteric binding site. ML254 is highly selective for mGlu5 versus other mGlu receptors, has a clean ancillary Ricerca profile, and suitable dystrophia myotonica protein kinase (DMPK) properties for systemic dosing in rodents. |
ターゲット&IC50 | mGluR5 (rat):8.03 nM (pEC50), mGluR5 (rat):9.3 nM (EC50) |
分子量 | 310.32 |
分子式 | C18H15FN2O2 |
CAS No. | 1428630-86-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 27.5 mg/mL (88.62 mM)
You can also refer to dose conversion for different animals. 詳細
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ML 254 1428630-86-7 Neuroscience GluR inhibit Inhibitor Metabotropic glutamate receptors mGluR ML-254 Schizophrenia ML254 inhibitor