Powder: -20°C for 3 years | In solvent: -80°C for 1 year
SB399885 (SB 399885) is an effective, brain penetrant, and orally active antagonist of SR-6. It shows 200-fold selectivity for SR-6 over other serotonin receptors (pKi: 9.11, 8.81, and 9.02 for human recombinant, native rat, and native human SR-6 receptors, respectively).
説明 | SB399885 (SB 399885) is an effective, brain penetrant, and orally active antagonist of SR-6. It shows 200-fold selectivity for SR-6 over other serotonin receptors (pKi: 9.11, 8.81, and 9.02 for human recombinant, native rat, and native human SR-6 receptors, respectively). |
ターゲット&IC50 | SR6 (human recombinant):9.11 (pKi), SR6 (native rat):8.81 (pKi), SR6 (native human):9.02 (pKi) |
別名 | SB399885 Hydrochloride, SB 399885, SB399885, SB-399885 |
分子量 | 446.35 |
分子式 | C18H21Cl2N3O4S |
CAS No. | 402713-80-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/ml (123.22 mM)
You can also refer to dose conversion for different animals. 詳細
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SB399885 402713-80-8 GPCR/G Protein Neuroscience 5-HT Receptor SB399885 Hydrochloride SB 399885 SB399885 HCl SB-399885 SB 399885 Hydrochloride SB-399885 HCl SB-399885 Hydrochloride Inhibitor inhibitor inhibit